SCHEMBL8328260

SCHEMBL8328260

O=C(O)CC1CCCc2cc(NC(=O)Cc3nc4ccccc4[nH]3)ccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.50
TDP1 Q9NUW8 2/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
POLB P06746 2/20 0.50
MAPT P10636 3/20 0.48
LMNA P02545 1/20 0.48
KDM4E B2RXH2 3/20 0.45
HPGD P15428 1/20 0.45
HSD17B10 Q99714 1/20 0.45
USP2 O75604 1/20 0.44
ITGB3 P05106 1/20 0.42
ITGAV P06756 1/20 0.42
LDLR P01130 1/20 0.42
CACNA1G O43497 1/20 0.42
HTT P42858 1/20 0.42
MMP2 P08253 1/20 0.42
MMP9 P14780 1/20 0.42
MMP8 P22894 1/20 0.42
MMP13 P45452 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8323660 0.80 ITGB3 (0.59) KMT2APOLBMAPTITGB3ITGAV
SCHEMBL7335166 0.77 ITGB3 (0.49) ALDH1A1TDP1MEN1KMT2APOLB
SCHEMBL7437624 0.77 ALDH1A1 (0.48) ALDH1A1TDP1MEN1KMT2APOLB
SCHEMBL15685943 0.74 ALDH1A1 (0.74) ALDH1A1TDP1MEN1KMT2APOLB
SCHEMBL7437616 0.70 ALDH1A1 (0.51) ALDH1A1TDP1MEN1KMT2APOLB
SCHEMBL8326108 0.69 ALDH1A1 (0.53) ALDH1A1TDP1MEN1KMT2APOLB
SCHEMBL30301824 0.67 FFAR1 (0.52) ALDH1A1MEN1KMT2AHPGDHTT
SCHEMBL3590904 0.67 FFAR1 (0.52) ALDH1A1MEN1KMT2AHPGDHTT
SCHEMBL761148 0.66 CHRM1 (0.71) ALDH1A1TDP1KMT2APOLBMAPT
SCHEMBL3450068 0.66 ESR1 (0.62)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869787-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-03-24 EP claimed
EP-0869787-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-14 EP claimed
WO-1997024119-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO claimed
EP-0869787-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-03-24 EP disclosed
EP-0869787-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-14 EP disclosed
WO-1997024119-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed