SCHEMBL8328885

SCHEMBL8328885

CCCCC(C(=O)O)=C(Nc1cccc(C(=O)OC)c1)C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.54
ALDH1A1 P00352 5/20 0.53
HPGD P15428 2/20 0.53
CYP1A2 P05177 2/20 0.53
CYP2C9 P11712 2/20 0.53
CYP2C19 P33261 2/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
NPC1 O15118 3/20 0.52
MDH1 P40925 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.49
MAPT P10636 2/20 0.47
TP53 P04637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7835265 0.85 RAB9A (0.56) RAB9AALDH1A1HPGDNPC1SMN1; SMN2
SCHEMBL8410515 0.82 RAB9A (0.55) RAB9AALDH1A1HPGDCYP1A2CYP2C9
SCHEMBL8410518 0.82 RAB9A (0.55) RAB9AALDH1A1HPGDCYP1A2CYP2C9
SCHEMBL7575475 0.82 ALDH1A1 (0.70) RAB9AALDH1A1HPGDCYP1A2CYP2C9
SCHEMBL7823722 0.81 MEN1 (0.55) ALDH1A1HPGDCYP2C19SMN1; SMN2MAPT
SCHEMBL7836111 0.79 MEN1 (0.56) RAB9AALDH1A1HPGDCYP1A2CYP2C9
SCHEMBL21998681 0.77 ALDH1A1 (0.67) RAB9AALDH1A1HPGDCYP1A2CYP2C9
SCHEMBL21998673 0.77 ALDH1A1 (0.67) RAB9AALDH1A1HPGDCYP1A2CYP2C9
SCHEMBL21998663 0.77 ALDH1A1 (0.67) RAB9AALDH1A1HPGDCYP1A2CYP2C9
SCHEMBL25933608 0.73 HTR7 (0.58) RAB9AALDH1A1HPGDCYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0498721-B1 N-substituted quinoline derivatives, process for their preparation, their use as pharmaceuticals and pharmaceutical compositions containing them HOECHST MARION ROUSSEL INC (FR) 1999-12-22 EP disclosed
EP-0498721-A1 N-substituted quinoline derivatives, process for their preparation, intermediates obtained, their use as pharmaceuticals and pharmaceutical compositions containing them ROUSSEL UCLAF (FR) 1992-08-12 EP disclosed