SCHEMBL8328601

SCHEMBL8328601

CNC(NC1CN(Cc2ccc(F)cc2)C1)=C(C#N)C#N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.41
ACHE P22303 2/20 0.41
BACE1 P56817 2/20 0.41
SIGMAR1 Q99720 4/20 0.39
DRD2 P14416 4/20 0.38
DRD4 P21917 1/20 0.38
FAAH O00519 1/20 0.38
ALDH1A1 P00352 2/20 0.38
PRKAA2 P54646 1/20 0.38
DRD3 P35462 3/20 0.38
CCR3 P51677 1/20 0.38
S1PR5 Q9H228 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
MCHR1 Q99705 2/20 0.37
MLNR O43193 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CHRM1 P11229 1/20 0.37
HTR2A P28223 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8329414 0.89 SIGMAR1 (0.53) BCHEACHEBACE1SIGMAR1ALDH1A1
SCHEMBL7491968 0.80 OPRK1 (0.44) DRD3CCR3
SCHEMBL8326114 0.77 MEN1 (0.48)
SCHEMBL8328838 0.77 MAPK1 (0.50) ACHEDRD4FAAH
SCHEMBL8326334 0.76 KMT2A (0.56) BCHEALDH1A1CCR3LMNAMCHR1
SCHEMBL7488935 0.76 DRD3 (0.51) SIGMAR1DRD2DRD4DRD3CCR3
SCHEMBL8329774 0.73 MAPK1 (0.48) FAAH
SCHEMBL8328605 0.71 BCHE (0.43) BCHEACHEBACE1DRD2DRD4
SCHEMBL8624159 0.71 BCHE (0.40) BCHEACHEBACE1DRD2FAAH
SCHEMBL8325591 0.70 OPRM1 (0.40) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5753654-A GASTROINTESTINAL DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-05-19 US disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760362-A1 NOVEL DIAMINOMETHYLIDENE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed