SCHEMBL8329466

SCHEMBL8329466

Cn1c(NCCC(COCc2ccccc2)NCc2ccc(F)cc2)c(C#N)c(=N)n(C)c1=S

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NRP1 O14786 1/20 0.33
LRRK2 Q5S007 1/20 0.32
CTSL P07711 1/20 0.30
CTSB P07858 1/20 0.30
CTSS P25774 1/20 0.30
GRM1 Q13255 2/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
TP53 P04637 1/20 0.30
GAA P10253 1/20 0.30
ALOX15 P16050 1/20 0.30
TSHR P16473 1/20 0.30
MAPK1 P28482 1/20 0.30
HSD17B10 Q99714 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
CASR P41180 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8322051 0.78 ALDH1A1 (0.42) LRRK2CTSLGRM1KDM4EALDH1A1
SCHEMBL8330575 0.77 MEN1 (0.35) KDM4EALDH1A1TP53GAAMAPK1
SCHEMBL8324185 0.76 CHRM2 (0.39) KDM4EALDH1A1TP53GAAMAPK1
SCHEMBL8328869 0.76 CHRM2 (0.44) KDM4EALDH1A1TP53GAAL3MBTL1
SCHEMBL8329010 0.76 CHRM2 (0.41) CTSLKDM4EALDH1A1TP53GAA
SCHEMBL8325662 0.75 CHRM2 (0.46) KDM4EALDH1A1TP53GAAL3MBTL1
SCHEMBL8326703 0.71 PLA2G1B (0.38) CTSLCTSBCTSSALDH1A1TSHR
SCHEMBL8323561 0.71 CTSS (0.35) CTSLCTSBCTSSALDH1A1L3MBTL1
SCHEMBL13995922 0.70 TACR1 (0.41) KDM4EALDH1A1L3MBTL1MEN1KMT2A
SCHEMBL8323557 0.70 LMNA (0.35) CTSLCTSBCTSSKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed