SCHEMBL8329759

SCHEMBL8329759

O=CC(CN1CCC(CO)CC1)NC(=O)OCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 1/20 0.48
CASP1 P29466 5/20 0.46
OPRK1 P41145 3/20 0.45
BCHE P06276 3/20 0.44
ACHE P22303 3/20 0.44
CACNA1F O60840 1/20 0.44
CACNA1D Q01668 1/20 0.44
CACNA1S Q13698 1/20 0.44
CACNA1C Q13936 1/20 0.44
CCR1 P32246 1/20 0.43
PREP P48147 2/20 0.42
PSMB1 P20618 1/20 0.42
PSMB5 P28074 1/20 0.42
PSMB2 P49721 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CYP1A2 P05177 1/20 0.42
MAOB P27338 1/20 0.42
TGM2 P21980 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24447908 0.79 CTSL (0.50) CASP1PSMB1PSMB5PSMB2ALDH1A1
SCHEMBL8138447 0.79 CTSL (0.50) CASP1PSMB1PSMB5PSMB2ALDH1A1
SCHEMBL7298029 0.77 CTRB1 (0.54) PSMB1PSMB5PSMB2
SCHEMBL13173061 0.77 CTRB1 (0.54) PSMB1PSMB5PSMB2
SCHEMBL8239267 0.77 CTRB1 (0.54) PSMB1PSMB5PSMB2
SCHEMBL3330029 0.77 CTSB (0.52) PSMB1PSMB5PSMB2ALDH1A1CYP1A2
SCHEMBL7271134 0.76 CTSL (0.56) CASP1ALDH1A1CYP1A2
SCHEMBL7271139 0.76 CTSL (0.56) CASP1ALDH1A1CYP1A2
SCHEMBL4425695 0.76 CASP1 (0.55) CASP1PSMB1PSMB5PSMB2
SCHEMBL1690791 0.76 CASP1 (0.55) CASP1PSMB1PSMB5PSMB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6002009-A Di-substituted 1,4-piperidine esters and amides having 5-HT4 antagonistic activity BOEHRINGER INGELHEIM ITALIA, S.P.A. (IT) 1999-12-14 US disclosed