SCHEMBL8328376

SCHEMBL8328376

COC(CN(Cc1ccc(F)cc1)C(=O)OC(C)(C)C)CN1C(=O)c2ccccc2C1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
KMT2A Q03164 2/20 0.38
RAB9A P51151 2/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
ALDH1A1 P00352 4/20 0.38
HSD17B10 Q99714 1/20 0.38
POLB P06746 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
GAA P10253 1/20 0.36
NR1H4 Q96RI1 1/20 0.36
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19545291 0.88 MAPK1 (0.43) CASP3SMN1; SMN2KMT2ARAB9AMEN1
SCHEMBL8329333 0.81 KDM1A (0.40) HDAC3HDAC1HDAC2NCOR2POLB
SCHEMBL8330600 0.80 KDM1A (0.39) HDAC3HDAC1HDAC2NCOR2MAPT
SCHEMBL31341735 0.80 GAA (0.42) CASP3KMT2ARAB9AMEN1NPC1
SCHEMBL8329022 0.80 ALDH1A1 (0.50) SMN1; SMN2KMT2AALDH1A1HSD17B10POLB
SCHEMBL8325503 0.80 SMN1; SMN2 (0.46) CASP3SMN1; SMN2KMT2ARAB9AMEN1
SCHEMBL8326721 0.79 MAOB (0.49) KMT2AALDH1A1HSD17B10POLB
SCHEMBL8326801 0.78 ACHE (0.50) KMT2AALDH1A1HSD17B10
SCHEMBL8330108 0.77 NPC1 (0.45) SMN1; SMN2KMT2ARAB9AMEN1NPC1
SCHEMBL8323152 0.76 KDM1A (0.37) CASP3RAB9ANPC1HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed