SCHEMBL8336582

SCHEMBL8336582

CC(c1ccc(-c2ccc(Br)cc2)cc1)c1c(O)c2ccccc2oc1=O

nearest known ligand 0.74

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
VKORC1 Q9BQB6 2/20 0.74
THRB P10828 1/20 0.67
NQO1 P15559 6/20 0.63
CYP2C9 P11712 6/20 0.60
CRHBP P24387 1/20 0.60
CASP7 P55210 1/20 0.60
CASP6 P55212 1/20 0.60
CRHR2 Q13324 1/20 0.60
HIF1A Q16665 1/20 0.60
TOP1 P11387 1/20 0.59
TOP2A P11388 1/20 0.57
KDM4E B2RXH2 1/20 0.56
POLB P06746 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8469143 0.90 VKORC1 (0.78) VKORC1NQO1CYP2C9CRHBPCASP7
SCHEMBL8334288 0.89 VKORC1 (0.76) VKORC1NQO1CYP2C9CRHBPCASP7
SCHEMBL8336015 0.88 THRB (0.64) VKORC1THRBNQO1CYP2C9CRHBP
SCHEMBL8336100 0.88 VKORC1 (0.74) VKORC1NQO1CYP2C9CRHBPCASP7
SCHEMBL8335244 0.86 THRB (0.78) VKORC1THRBNQO1CYP2C9CRHBP
SCHEMBL8337124 0.85 CYP2C9 (0.77) VKORC1THRBNQO1CYP2C9TOP1
SCHEMBL8334704 0.85 VKORC1 (0.70) VKORC1NQO1CYP2C9CRHBPCASP7
SCHEMBL7349603 0.85 VKORC1 (1.00) VKORC1NQO1CYP2C9CRHBPCASP7
SCHEMBL8523615 0.85 THRB (0.70) VKORC1THRBNQO1CYP2C9KDM4E
SCHEMBL8335689 0.84 VKORC1 (0.69) VKORC1NQO1CYP2C9CRHBPCASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999001446-A1 NOVEL 4-HYDROXY-2H-1-(THIO)PYRAN-2-ONES DERIVATIVES AND THEIR USE AS RAT POISON LIPHATEC (FR) 1999-01-14 WO disclosed