SCHEMBL8335106

SCHEMBL8335106

Cc1ccc(CNC(=O)c2cc(C(=O)NCc3ccc4c(c3)OCCO4)ncn2)o1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 3/20 0.50
ALDH1A1 P00352 3/20 0.50
HPGD P15428 5/20 0.49
MAPK1 P28482 1/20 0.49
POLB P06746 2/20 0.47
NPC1 O15118 3/20 0.47
RAB9A P51151 2/20 0.47
PKM P14618 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
CHRM4 P08173 1/20 0.46
HTT P42858 2/20 0.45
MEN1 O00255 1/20 0.45
USP2 O75604 1/20 0.45
ESR1 P03372 1/20 0.45
KMT2A Q03164 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HSD17B10 Q99714 3/20 0.45
KDM4E B2RXH2 2/20 0.45
LMNA P02545 1/20 0.45
TP53 P04637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14602312 0.89 RAB9A (0.55) MMP13HPGDMAPK1POLBNPC1
SCHEMBL8348338 0.81 MMP13 (0.78) MMP13ALDH1A1HPGDPOLBPKM
SCHEMBL5617718 0.81 ALDH1A1 (0.52) MMP13ALDH1A1HPGDMAPK1NPC1
SCHEMBL8349714 0.79 MMP13 (0.61) MMP13ALDH1A1HPGDPOLBPKM
SCHEMBL8360152 0.78 KMT2A (0.53) MMP13ALDH1A1HPGDMAPK1NPC1
SCHEMBL8335113 0.78 SMN1; SMN2 (0.64) MMP13ALDH1A1HPGDMAPK1NPC1
SCHEMBL8335466 0.78 MMP13 (0.72) MMP13ALDH1A1HPGDMAPK1POLB
SCHEMBL4716678 0.76 ALDH1A1 (0.54) ALDH1A1HPGDMAPK1POLBNPC1
SCHEMBL8335066 0.76 MMP13 (0.53) MMP13ALDH1A1HPGDMAPK1NPC1
SCHEMBL8336049 0.75 MMP13 (0.52) MMP13ALDH1A1HPGDMAPK1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7166609-B2 Pyrimidine-4,6-dicarboxylic acid diamides for selectively inhibiting collagenases SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2007-01-23 US disclosed
US-7166609-B2 Pyrimidine-4,6-dicarboxylic acid diamides for selectively inhibiting collagenases SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2007-01-23 US disclosed
WO-2004041788-A1 NOVEL PYRIMIDINE-4,6-DICARBOXAMIDES FOR THE SELECTIVE INHIBITION OF COLLAGENASES AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2004-05-21 WO disclosed