SCHEMBL8335176

SCHEMBL8335176

C#Cc1c(C(=O)O)cccc1-c1ccc2c(c1)C(c1ccc(C(C)(C)C)cc1)=CC(C)(C)O2

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RARB P10826 5/20 0.41
RARA P10276 4/20 0.41
RARG P13631 4/20 0.41
PPARG P37231 1/20 0.34
PPARA Q07869 1/20 0.33
AKR1C2 P52895 1/20 0.32
AKR1C1 Q04828 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPK1 P28482 1/20 0.32
GFER P55789 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
RORB Q92753 1/20 0.31
DHODH Q02127 1/20 0.31
OPRD1 P41143 1/20 0.31
TRPV1 Q8NER1 2/20 0.30
RXRA P19793 1/20 0.30
RXRB P28702 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8332455 0.91 RARA (0.44) RARBRARARARGPPARGPPARA
SCHEMBL8331802 0.89 RARA (0.52) RARBRARARARGPPARGOPRD1
SCHEMBL8331104 0.88 RARA (0.41) RARBRARARARGPPARGPPARA
SCHEMBL8329425 0.87 RARA (0.41) RARBRARARARGDHODHOPRD1
SCHEMBL8331248 0.81 RARB (0.38) RARBRARARARGAKR1C2AKR1C1
SCHEMBL8335170 0.77 RARB (0.44) RARBRARARARGPPARGPPARA
SCHEMBL6594110 0.73 RARB (0.60) RARBRARARARGRXRARXRB
SCHEMBL24727636 0.73 RARB (0.52) RARBRARARARGOPRD1RXRA
SCHEMBL8335174 0.70 RARB (0.42) RARBRARARARGPPARGPPARA
SCHEMBL12365151 0.66 RARA (0.63) RARBRARARARGOPRD1RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5958954-A 2,2-DIALKYL-4-ARYL-SUBSTITUTED BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES ALLERGAN SALES, INC. (US) 1999-09-28 US disclosed