SCHEMBL8336015

SCHEMBL8336015

CC(C)C(c1ccc(-c2ccc(Br)cc2)cc1)c1c(O)c2ccccc2oc1=O

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.64
NQO1 P15559 11/20 0.64
CYP2C9 P11712 2/20 0.60
CRHBP P24387 1/20 0.60
CASP7 P55210 1/20 0.60
CASP6 P55212 1/20 0.60
CRHR2 Q13324 1/20 0.60
HIF1A Q16665 1/20 0.60
TOP1 P11387 1/20 0.60
TOP2A P11388 1/20 0.58
KDM4E B2RXH2 1/20 0.57
POLB P06746 1/20 0.57
VKORC1 Q9BQB6 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7362123 0.96 NQO1 (0.64) THRBNQO1CYP2C9CRHBPCASP7
SCHEMBL8336582 0.88 VKORC1 (0.74) THRBNQO1CYP2C9CRHBPCASP7
SCHEMBL7355322 0.86 VKORC1 (0.74) NQO1CYP2C9CRHBPCASP7CASP6
SCHEMBL8335244 0.84 THRB (0.78) THRBNQO1CYP2C9CRHBPCASP7
SCHEMBL12028810 0.83 NQO1 (0.86) NQO1CYP2C9CRHBPCASP7CASP6
SCHEMBL8337124 0.83 CYP2C9 (0.77) THRBNQO1CYP2C9TOP1KDM4E
SCHEMBL8523615 0.83 THRB (0.70) THRBNQO1CYP2C9KDM4EPOLB
SCHEMBL8332272 0.81 THRB (0.71) THRBNQO1CYP2C9KDM4EVKORC1
SCHEMBL8333320 0.81 THRB (0.70) THRBNQO1CYP2C9TOP1TOP2A
SCHEMBL8334663 0.80 THRB (0.72) THRBNQO1CYP2C9TOP1TOP2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999001446-A1 NOVEL 4-HYDROXY-2H-1-(THIO)PYRAN-2-ONES DERIVATIVES AND THEIR USE AS RAT POISON LIPHATEC (FR) 1999-01-14 WO disclosed