SCHEMBL8337229

SCHEMBL8337229

NC(=O)c1cc(Br)ccc1OCc1ccc(C(F)(F)F)cc1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.53
PTPN1 P18031 2/20 0.52
PTGER1 P34995 2/20 0.51
RXRA P19793 1/20 0.49
RXRB P28702 1/20 0.49
RXRG P48443 1/20 0.49
MRGPRX4 Q96LA9 3/20 0.47
CCR5 P51681 3/20 0.47
LRRK2 Q5S007 3/20 0.46
PARP1 P09874 2/20 0.46
LMNA P02545 2/20 0.44
HTT P42858 1/20 0.44
POLB P06746 1/20 0.44
PARP2 Q9UGN5 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8337276 0.85 PTGER1 (0.49) MAOBPTGER1MRGPRX4CCR5LRRK2
SCHEMBL4723723 0.82 LRRK2 (0.58) CCR5LRRK2PARP1LMNAPOLB
SCHEMBL8337852 0.80 PTGES (0.59) CCR5LRRK2PARP1
SCHEMBL8336987 0.79 LRRK2 (0.53) CCR5LRRK2PARP1LMNAPOLB
SCHEMBL8337376 0.79 MEN1 (0.54) PTGER1CCR5LRRK2PARP1LMNA
SCHEMBL8243758 0.76 LRRK2 (0.58) PTPN1PTGER1RXRARXRBRXRG
SCHEMBL5699854 0.76 PTPN1 (0.64) PTPN1PTGER1RXRARXRBRXRG
SCHEMBL30679655 0.76 PTPN1 (0.64) PTPN1PTGER1RXRARXRBRXRG
SCHEMBL27522244 0.76 MAOB (0.52) MAOBPTGER1RXRARXRBRXRG
SCHEMBL856030 0.75 RXRA (0.70) MAOBPTPN1RXRARXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014844-A2 ARYL AND HETEROARYL COMPOUNDS AND METHODS TO MODULATE COAGULATION TRANSTECH PHARMA, INC. (US) 2004-02-19 WO disclosed