SCHEMBL8338491

SCHEMBL8338491

[c]1cccc(C2NCCO2)c1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
SLC6A2 P23975 1/20 0.42
ADRA1A P35348 1/20 0.42
HTR2B P41595 1/20 0.42
SLC6A3 Q01959 1/20 0.42
CHRNA7 P36544 1/20 0.36
DRD3 P35462 2/20 0.31
DRD2 P14416 1/20 0.31
TACR1 P25103 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8117490 0.79 ALDH1A1 (0.47) ALDH1A1SLC6A2ADRA1AHTR2BSLC6A3
SCHEMBL2257666 0.79 SLC6A2 (0.58) ALDH1A1SLC6A2ADRA1AHTR2BSLC6A3
SCHEMBL460150 0.79 SLC6A2 (0.58) ALDH1A1SLC6A2ADRA1AHTR2BSLC6A3
SCHEMBL594796 0.77 ALDH1A1 (0.57) ALDH1A1SLC6A2ADRA1AHTR2BSLC6A3
SCHEMBL1023795 0.76 ALDH1A1 (0.59) ALDH1A1SLC6A2ADRA1AHTR2BSLC6A3
SCHEMBL1492682 0.72 DRD2 (0.56) DRD3DRD2
SCHEMBL4900607 0.71 MEN1 (0.38)
SCHEMBL8572944 0.70 ALDH1A1 (0.50) ALDH1A1SLC6A2ADRA1AHTR2BSLC6A3
SCHEMBL5172003 0.70 CHRNB2 (0.56) ALDH1A1SLC6A2ADRA1AHTR2BSLC6A3
SCHEMBL7215080 0.70 ALDH1A1 (0.50) ALDH1A1SLC6A2ADRA1AHTR2BSLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5877312-A Method for preparing alkylating agents for their use for alkylating cyclic ureas DUPONT PHARMACEUTICALS COMPANY (US) 1999-03-02 US claimed
US-5637780-A Method for preparing alkylating agents and their use for alkylating cyclic ureas THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-06-10 US claimed
EP-0767770-A1 METHOD FOR PREPARING ALKYLATING AGENTS AND THEIR USE FOR ALKYLATING CYCLIC UREAS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-04-16 EP claimed
WO-1996000708-A1 METHOD FOR PREPARING ALKYLATING AGENTS AND THEIR USE FOR ALKYLATING CYCLIC UREAS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-01-11 WO claimed
US-5877312-A Method for preparing alkylating agents for their use for alkylating cyclic ureas DUPONT PHARMACEUTICALS COMPANY (US) 1999-03-02 US disclosed
US-5637780-A Method for preparing alkylating agents and their use for alkylating cyclic ureas THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-06-10 US disclosed
EP-0767770-A1 METHOD FOR PREPARING ALKYLATING AGENTS AND THEIR USE FOR ALKYLATING CYCLIC UREAS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-04-16 EP disclosed
WO-1996000708-A1 METHOD FOR PREPARING ALKYLATING AGENTS AND THEIR USE FOR ALKYLATING CYCLIC UREAS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-01-11 WO disclosed