SCHEMBL8343301

SCHEMBL8343301

Cc1cccc(C(F)(F)Br)c1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.42
GABRA1 P14867 1/20 0.39
GABRB2 P47870 1/20 0.39
ACHE P22303 3/20 0.37
CYP1A2 P05177 1/20 0.35
CYP2A6 P11509 1/20 0.35
TRPA1 O75762 2/20 0.34
ATM Q13315 1/20 0.34
ALDH1A1 P00352 2/20 0.33
CA2 P00918 2/20 0.33
CA1 P00915 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
HSD11B1 P28845 1/20 0.33
TSHR P16473 1/20 0.33
MPL P40238 1/20 0.33
P2RX7 Q99572 1/20 0.32
PDK2 Q15119 2/20 0.31
SCN8A Q9UQD0 1/20 0.30
PDK1 Q15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL476650 0.84 MPL (0.44) KIF11GABRA1GABRB2ACHECYP1A2
SCHEMBL9882817 0.82 GABRA1 (0.43) KIF11GABRA1GABRB2ACHECYP1A2
SCHEMBL8846936 0.80 KIF11 (0.41) KIF11GABRA1GABRB2ACHECYP1A2
SCHEMBL9626868 0.79 GABRA1 (0.56) KIF11GABRA1GABRB2ACHECYP1A2
SCHEMBL28574005 0.77 P2RX7 (0.36) CYP1A2CYP2A6HSD11B1TSHRMPL
SCHEMBL25078710 0.77 KIF11 (0.40) KIF11GABRA1GABRB2ACHECYP1A2
SCHEMBL4002333 0.76 HSD11B1 (0.39) HSD11B1MPLP2RX7PDK2
SCHEMBL30018336 0.76 KIF11 (0.45) KIF11GABRA1GABRB2ACHECYP1A2
SCHEMBL23886233 0.76 KIF11 (0.45) KIF11GABRA1GABRB2ACHECYP1A2
SCHEMBL23344925 0.75 KIF11 (0.39) KIF11GABRA1GABRB2ACHECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114616232-A Azepadinopyrimidine derivatives and medical application thereof 正大天晴药业集团南京顺欣制药有限公司 2022-06-10 CN disclosed
WO-1999011612-A2 SUBSTITUTED CYCLIC COMPOUNDS AND MIXTURES COMPRISING SAME ISIS PHARMACEUTICALS, INC. (US) 1999-03-11 WO disclosed