SCHEMBL8347170

SCHEMBL8347170

CC(C)c1nc(CCC(=O)O)n(Cc2ccncc2)c1Sc1cccc(F)c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 2/20 0.42
ENPP2 Q13822 6/20 0.39
LMNA P02545 3/20 0.38
RXFP1 Q9HBX9 1/20 0.37
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
TP53 P04637 1/20 0.34
SLC6A9 P48067 2/20 0.34
ALDH1A1 P00352 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
GSK3B P49841 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8343038 0.92 TBXA2R (0.42) TBXA2RENPP2LMNARXFP1ALDH1A1
SCHEMBL8344845 0.90 PKM (0.41) TBXA2RENPP2LMNARXFP1GRIN1
SCHEMBL6968454 0.90 ENPP2 (0.39) TBXA2RENPP2LMNAGRIN1GRIN2B
SCHEMBL6967782 0.90 LMNA (0.39) TBXA2RENPP2LMNARXFP1TP53
SCHEMBL8347165 0.90 LMNA (0.45) TBXA2RENPP2LMNARXFP1MEN1
SCHEMBL6975612 0.89 GRIN1 (0.35) ENPP2LMNAGRIN1GRIN2BTP53
SCHEMBL7085890 0.87 GSK3B (0.34) ENPP2LMNAGRIN1GRIN2BTP53
SCHEMBL6975055 0.87 GRIN1 (0.35) ENPP2LMNAGRIN1GRIN2BTP53
SCHEMBL6975545 0.87 GRIN1 (0.34) ENPP2LMNAGRIN1GRIN2BTP53
SCHEMBL8345427 0.87 TBXA2R (0.37) TBXA2RSLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed