SCHEMBL8350434

SCHEMBL8350434

Cc1onc(-c2cccc(F)c2)c1NS(=O)(=O)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
NPSR1 Q6W5P4 1/20 0.50
MT-CO2 P00403 2/20 0.47
PTGS2 P35354 2/20 0.47
TSHR P16473 1/20 0.47
MAPK1 P28482 1/20 0.47
EDNRB P24530 5/20 0.46
EDNRA P25101 5/20 0.46
PKM P14618 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
MAP2K7 O14733 1/20 0.44
MAP2K4 P45985 1/20 0.44
KAT6A Q92794 1/20 0.44
PTPN1 P18031 1/20 0.43
PTPN5 P54829 1/20 0.43
GPBAR1 Q8TDU6 1/20 0.43
FFAR4 Q5NUL3 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8474183 0.90 ALDH1A1 (0.49) ALDH1A1NPSR1MT-CO2PTGS2TSHR
SCHEMBL6435523 0.87 ALDH1A1 (0.63) ALDH1A1NPSR1MT-CO2PTGS2TSHR
SCHEMBL8477494 0.87 ALDH1A1 (0.46) ALDH1A1NPSR1MT-CO2PTGS2TSHR
SCHEMBL8473859 0.86 PTGS2 (0.53) ALDH1A1NPSR1MT-CO2PTGS2TSHR
SCHEMBL8475736 0.85 ALDH1A1 (0.59) ALDH1A1NPSR1MT-CO2PTGS2TSHR
SCHEMBL8473536 0.85 ALDH1A1 (0.47) ALDH1A1NPSR1MT-CO2PTGS2TSHR
Benzenesulfonamide SCHEMBL7180310 0.81 PTGS2 (0.62) ALDH1A1NPSR1MT-CO2PTGS2TSHR
SCHEMBL8477521 0.81 ALDH1A1 (0.58) ALDH1A1NPSR1MT-CO2PTGS2TSHR
SCHEMBL6169842 0.81 PTGS2 (0.47) ALDH1A1NPSR1MT-CO2PTGS2TSHR
SCHEMBL8476183 0.81 KMO (0.51) ALDH1A1NPSR1MT-CO2PTGS2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5932598-A NOVEL SUBSTITUTED SULFONAMIDE COMPOUNDS USEFUL AS PRODRUGS; ADMINISTERING TO TREAT INFLAMMATION-ASSOCIATED PAIN DUE TO CANCER, DENTAL PAIN; CYCLOOXYGENASE-2 INHIBITORS G. D. SEARLE & CO. (US) 1999-08-03 US disclosed
US-5859257-A ANTIINFLAMMATORY, ANTIARTHRITIC AGENTS G. D. SEARLE & CO. (US) 1999-01-12 US disclosed