SCHEMBL8350460

SCHEMBL8350460

COc1cc(C(=O)N2CCC(c3cccs3)C2)cc(OC)c1OC

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.59
MEN1 O00255 1/20 0.59
KMT2A Q03164 1/20 0.59
UBE2M P61081 1/20 0.54
DCUN1D1 Q96GG9 1/20 0.54
CYP1A2 P05177 1/20 0.53
POLB P06746 1/20 0.51
GAA P10253 2/20 0.51
PDE4B Q07343 1/20 0.50
HTT P42858 2/20 0.49
KDM4E B2RXH2 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
PDE2A O00408 1/20 0.48
TSHR P16473 3/20 0.48
MAPK1 P28482 2/20 0.48
HSD17B10 Q99714 1/20 0.47
LMNA P02545 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8351152 0.81 ALDH1A1 (0.64) ALDH1A1MEN1KMT2AUBE2MDCUN1D1
SCHEMBL8636998 0.78 ALDH1A1 (0.65) ALDH1A1UBE2MDCUN1D1CYP1A2GAA
SCHEMBL8352641 0.78 PDE4B (0.65) GAAPDE4BKDM4ELMNA
SCHEMBL8351389 0.78 ALDH1A1 (0.56) ALDH1A1MEN1KMT2AUBE2MDCUN1D1
SCHEMBL8636740 0.78 ALDH1A1 (0.56) ALDH1A1MEN1KMT2AUBE2MDCUN1D1
SCHEMBL8638316 0.77 SCD5 (0.55) ALDH1A1MEN1KMT2AUBE2MDCUN1D1
SCHEMBL8638113 0.77 LMNA (0.60) ALDH1A1MEN1KMT2AUBE2MDCUN1D1
SCHEMBL8635894 0.77 PROKR1 (0.53) ALDH1A1MEN1KMT2AUBE2MDCUN1D1
SCHEMBL8638632 0.77 PDE4B (0.53) ALDH1A1MEN1KMT2AUBE2MDCUN1D1
SCHEMBL724938 0.76 ALDH1A1 (0.71) ALDH1A1MEN1KMT2AUBE2MDCUN1D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5861416-A TREATMENT OF ASTHMA OR COUGH MERRELL PHARMACEUTICALS INC. (US) 1999-01-19 US disclosed
US-5824690-A TREATING ASTHMA, COUGH HOECHST MARION ROUSSEL INC. (US) 1998-10-20 US disclosed