SCHEMBL8359252

SCHEMBL8359252

O=c1[nH]c2c(c3ccc(F)cc13)CN(CCCN1CCc3ccccc3C1)CC2

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.56
PARP1 P09874 2/20 0.53
ADRA1D P25100 1/20 0.51
ADRA1B P35368 1/20 0.51
HTR1A P08908 3/20 0.49
DRD2 P14416 3/20 0.49
HTR2A P28223 3/20 0.49
HTR7 P34969 3/20 0.49
DRD3 P35462 3/20 0.49
HTR2B P41595 3/20 0.49
APAF1 O14727 1/20 0.49
ACHE P22303 1/20 0.48
HRH1 P35367 2/20 0.47
SLC6A4 P31645 1/20 0.47
HTR5A P47898 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30029262 0.86 PARP1 (0.70) SIGMAR1PARP1APAF1ACHE
SCHEMBL8359243 0.86 PARP1 (0.75) PARP1HTR1ADRD2HTR2AHTR7
SCHEMBL8359382 0.81 ACHE (0.73) PARP1ACHE
SCHEMBL1719867 0.75 KDM4E (0.61) ADRA1DADRA1BHTR1ADRD2HTR2A
SCHEMBL8362890 0.73 PARP1 (0.76) SIGMAR1PARP1
SCHEMBL16335515 0.71 SIGMAR1 (0.68) SIGMAR1APAF1ACHE
SCHEMBL8363079 0.70 PARP1 (0.74) PARP1
SCHEMBL7529695 0.70 SLC6A4 (0.73) ADRA1DADRA1BHTR1ADRD2HTR2A
SCHEMBL8359236 0.69 PARP1 (1.00) PARP1
SCHEMBL14444052 0.69 PARP1 (0.76) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7247641-B2 Compounds, derivatives, compositions, preparation and uses MGI GP, INC. (US) 2007-07-24 US disclosed
US-7247641-B2 Compounds, derivatives, compositions, preparation and uses MGI GP, INC. (US) 2007-07-24 US disclosed
WO-2003014121-A9 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARM INC (US) 2004-03-25 WO disclosed
WO-2003014121-A1 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARMACEUTICALS INC. (US) 2003-02-20 WO disclosed