SCHEMBL8359382

SCHEMBL8359382

O=c1[nH]c2c(c3ccc(F)cc13)CN(Cc1ccccc1)CC2

nearest known ligand 0.73

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACHE P22303 4/20 0.73
HDAC1 Q13547 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
PARP1 P09874 1/20 0.54
GABRA1 P14867 4/20 0.54
GABRA2 P47869 4/20 0.54
GABRA5 P31644 1/20 0.54
GABRA3 P34903 1/20 0.54
SLC6A5 Q9Y345 1/20 0.54
AKR1B1 P15121 1/20 0.53
HTR6 P50406 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8359258 0.87 ACHE (0.71) ACHEHDAC1HDAC6PARP1GABRA1
SCHEMBL8359525 0.86 ACHE (0.73) ACHEHDAC1HDAC6GABRA1GABRA2
SCHEMBL8359252 0.81 SIGMAR1 (0.56) ACHEPARP1
SCHEMBL30029262 0.79 PARP1 (0.70) ACHEPARP1
SCHEMBL2625346 0.78 SLC6A5 (0.80) ACHEGABRA1GABRA2SLC6A5AKR1B1
SCHEMBL8359307 0.77 SLC6A5 (0.74) ACHEHDAC1HDAC6PARP1SLC6A5
SCHEMBL633048 0.74 ACHE (1.00) ACHEHDAC1HDAC6AKR1B1
SCHEMBL29915094 0.74 SLC6A5 (0.61) ACHEHDAC1HDAC6SLC6A5
SCHEMBL27002308 0.74 SLC6A5 (0.61) ACHEHDAC1HDAC6SLC6A5
SCHEMBL8359419 0.73 PARP1 (0.74) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7247641-B2 Compounds, derivatives, compositions, preparation and uses MGI GP, INC. (US) 2007-07-24 US disclosed
US-7247641-B2 Compounds, derivatives, compositions, preparation and uses MGI GP, INC. (US) 2007-07-24 US disclosed
WO-2003014121-A9 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARM INC (US) 2004-03-25 WO disclosed
WO-2003014121-A1 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARMACEUTICALS INC. (US) 2003-02-20 WO disclosed