SCHEMBL8359307

SCHEMBL8359307

O=c1[nH]c2c(c3ccccc13)CCN(Cc1ccccc1)C2

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A5 Q9Y345 1/20 0.74
MEN1 O00255 3/20 0.58
KMT2A Q03164 3/20 0.58
ATM Q13315 2/20 0.58
GAA P10253 1/20 0.58
ACHE P22303 1/20 0.56
RCE1 Q9Y256 1/20 0.55
PARP1 P09874 5/20 0.54
HDAC1 Q13547 2/20 0.54
HDAC6 Q9UBN7 2/20 0.54
HDAC3 O15379 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC10 Q969S8 1/20 0.50
HDAC11 Q96DB2 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
HDAC9 Q9UKV0 1/20 0.50
HDAC5 Q9UQL6 1/20 0.50
HTR1A P08908 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8359258 0.89 ACHE (0.71) SLC6A5ACHEPARP1HDAC1HDAC6
SCHEMBL29915094 0.88 SLC6A5 (0.61) SLC6A5MEN1KMT2AATMGAA
SCHEMBL8360515 0.86 HTR1A (0.61) SLC6A5MEN1KMT2AATMGAA
SCHEMBL4144313 0.85 SLC6A5 (1.00) SLC6A5MEN1KMT2AATMGAA
SCHEMBL8363111 0.81 PARP1 (0.77) SLC6A5MEN1KMT2AGAAPARP1
SCHEMBL8360513 0.80 PARP1 (0.77) SLC6A5PARP1
SCHEMBL2344021 0.79 SLC6A5 (0.71) SLC6A5MEN1KMT2AATMGAA
SCHEMBL8359246 0.77 PARP1 (0.68) PARP1HDAC1HDAC6
SCHEMBL8359382 0.77 ACHE (0.73) SLC6A5ACHEPARP1HDAC1HDAC6
SCHEMBL8359525 0.77 ACHE (0.73) SLC6A5ACHEHDAC1HDAC6DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7247641-B2 Compounds, derivatives, compositions, preparation and uses MGI GP, INC. (US) 2007-07-24 US disclosed
US-7247641-B2 Compounds, derivatives, compositions, preparation and uses MGI GP, INC. (US) 2007-07-24 US disclosed
WO-2003014121-A9 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARM INC (US) 2004-03-25 WO disclosed
WO-2003014121-A1 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARMACEUTICALS INC. (US) 2003-02-20 WO disclosed