SCHEMBL8366182

SCHEMBL8366182

C=CCCC(=O)c1ccc(CC(NC(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C(=O)C(F)(F)CNCc2ccccc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSD P07339 3/20 0.43
CASP3 P42574 4/20 0.43
CASP1 P29466 3/20 0.43
CASP9 P55211 2/20 0.43
CASP7 P55210 2/20 0.41
LMNA P02545 1/20 0.39
CYP3A4 P08684 1/20 0.39
CAPN1 P07384 1/20 0.39
ELANE P08246 2/20 0.39
TACR1 P25103 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8361282 0.88 CTSD (0.47) CTSDCASP3CASP1CASP9CASP7
SCHEMBL8366184 0.82 CTSD (0.43) CTSDCASP3CASP1CASP9CASP7
SCHEMBL8366143 0.79 CTSD (0.45) CTSDCASP3CASP7
SCHEMBL8492203 0.77 CTSD (0.54) CTSDCASP3CASP7CAPN1ELANE
SCHEMBL7806370 0.73 CTSD (0.49) CTSDCASP3CASP7TACR1
SCHEMBL23234582 0.72 ALDH1A1 (0.59) CTSDCASP3CASP7CAPN1TACR1
SCHEMBL6269817 0.72 CTSD (0.59) CTSDCASP3CASP7TACR1
SCHEMBL8736216 0.72 CTSD (0.53) CTSD
SCHEMBL3058668 0.71 ECE1 (0.61) CTSDCASP3CASP7CAPN1TACR1
SCHEMBL25287172 0.71 ECE1 (0.61) CTSDCASP3CASP7CAPN1TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0717731-B1 DIFLUORO STATONE ANTIVIRAL ANALOGS MERRELL PHARMA INC (US) 1999-04-21 EP claimed