SCHEMBL8366184

SCHEMBL8366184

CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)NC(Cc1ccc(CCCC=C=O)cc1)C(=O)C(F)(F)CNCc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSD P07339 3/20 0.43
CA2 P00918 1/20 0.41
CA5A P35218 1/20 0.41
CASP3 P42574 3/20 0.41
CASP7 P55210 1/20 0.41
CASP1 P29466 2/20 0.40
TACR1 P25103 1/20 0.40
CASP9 P55211 1/20 0.40
CTSL P07711 3/20 0.40
CTSK P43235 2/20 0.40
CTSB P07858 1/20 0.40
CTSS P25774 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8361286 0.89 CTSD (0.47) CTSDCA2CA5ACASP3CASP7
SCHEMBL8366182 0.82 CTSD (0.43) CTSDCASP3CASP7CASP1TACR1
SCHEMBL8366143 0.79 CTSD (0.45) CTSDCASP3CASP7
SCHEMBL8492203 0.78 CTSD (0.54) CTSDCASP3CASP7TACR1CTSL
SCHEMBL7806370 0.74 CTSD (0.49) CTSDCA2CA5ACASP3CASP7
SCHEMBL7416124 0.74 CASP3 (0.49) CTSDCA2CASP3CASP7CASP1
SCHEMBL8736216 0.73 CTSD (0.53) CTSDCTSKCTSS
SCHEMBL7414133 0.72 CTSB (0.56) CASP3CTSLCTSKCTSBCTSS
SCHEMBL7420909 0.72 CTSB (0.56) CASP3CTSLCTSKCTSBCTSS
SCHEMBL7415829 0.72 CTSB (0.56) CASP3CTSLCTSKCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0717731-B1 DIFLUORO STATONE ANTIVIRAL ANALOGS MERRELL PHARMA INC (US) 1999-04-21 EP claimed