SCHEMBL8366284

SCHEMBL8366284

Cc1nnc(C2(c3ccccc3)CCN(OS(=O)(=O)c3ccccc3)CC2)o1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY1R P25929 1/20 0.42
PARL Q9H300 1/20 0.35
NR3C2 P08235 1/20 0.34
APLNR P35414 1/20 0.34
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.33
OPRM1 P35372 2/20 0.33
DRD4 P21917 1/20 0.33
ALDH1A1 P00352 2/20 0.33
MAPK1 P28482 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
GRIN1 Q05586 1/20 0.33
KCNH2 Q12809 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6544549 0.85 VDR (0.38) NPY1RNR3C2KMT2AMEN1ALDH1A1
SCHEMBL8367127 0.70 OPRD1 (0.56) NPY1RKMT2AMEN1OPRM1ALDH1A1
SCHEMBL3286704 0.69 PARL (0.60) PARLKMT2AMEN1ALDH1A1L3MBTL1
Water SCHEMBL6543265 0.68 BACE1 (0.43) KMT2AMEN1ALDH1A1KDM4EMAPT
SCHEMBL7749126 0.67 VDR (0.35) KMT2AMEN1OPRM1DRD4ALDH1A1
SCHEMBL7683426 0.67 POLB (0.46) PARLKMT2AMEN1ALDH1A1KCNH2
SCHEMBL28177660 0.66 PARL (0.56) PARLKMT2AMEN1ALDH1A1MAPK1
SCHEMBL1493760 0.66 PARL (0.56) PARLKMT2AMEN1ALDH1A1L3MBTL1
SCHEMBL27630329 0.66 PARL (0.49) PARLKMT2AMEN1ALDH1A1L3MBTL1
SCHEMBL9517665 0.66 TSHR (0.51) PARLKMT2AMEN1ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965580-A TREATMENT OF SUBSTANCE P- AND NEUROKININ-DEPENDENT DISORDERS SANOFI (FR) 1999-10-12 US disclosed
US-5939411-A PIPERIDINE DERIVATIVES SUBSTITUTED AT POSITION 4 WITH NEW FUNCTIONS OTHER THAN THOSE DESCRIBED PREVIOUSLY HAVE A HIGH AFFINITY FOR NEUROKININ RECEPTORS AND ARE USEFUL FOR TREATMENT OF SUBSTANCE P AND NEUROKININ DEPENDENT PATHOLOGIES SANOFI (FR) 1999-08-17 US disclosed
US-5830906-A Piperidine derivatives, process for obtaining them and pharmaceutical compositions containing them SANOFI (FR) 1998-11-03 US disclosed