SCHEMBL8375699

SCHEMBL8375699

CC(C)(C)ON(C=O)CCOc1cc(-c2cccc3ccccc23)on1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 1/20 0.33
S1PR1 P21453 1/20 0.33
S1PR3 Q99500 1/20 0.33
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33
HTR1B P28222 2/20 0.32
HTR2C P28335 1/20 0.32
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TP53 P04637 1/20 0.31
GLA P06280 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
MAPK1 P28482 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8377369 0.87 NPC1 (0.34) SLC6A9NPC1ALDH1A1MAPTHPGD
SCHEMBL8377377 0.86 NPC1 (0.38) NPC1ALDH1A1MAPTHPGDRAB9A
SCHEMBL8377399 0.85 ALDH1A1 (0.44) KDM4ENPC1ALDH1A1GAAMAPT
SCHEMBL8375001 0.84 NR1H2 (0.31) NPC1RAB9A
SCHEMBL8380161 0.84 NR1H2 (0.36) KDM4ENPC1RAB9ASMN1; SMN2TDP1
SCHEMBL8378946 0.83 CXCR1 (0.40) ALDH1A1
SCHEMBL8376838 0.81 NR1H4 (0.32) MAPT
SCHEMBL8380155 0.79 ACKR3 (0.36)
SCHEMBL8376904 0.79 ALOX15 (0.36) KDM4ENPC1ALDH1A1TP53MAPT
SCHEMBL8375555 0.78 NPC1 (0.35) S1PR1NPC1ALDH1A1TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6005116-A HAVE INHIBITION ACTIVITIES AGAINST TYPE A-MONOAMINE OXIDASE; TREATING OR PREVENTING DEPRESSION, PARKINSON'S DISEASE, ALZEHEIMER'S DEMENTIA, OR CEREBROVASCULAR DEMENTIA SANKYO COMPANY, LIMITED (JP) 1999-12-21 US disclosed
EP-0885891-A1 ISOXAZOLE DERIVATIVES SANKYO COMPANY LIMITED (JP) 1998-12-23 EP disclosed