SCHEMBL8377377

SCHEMBL8377377

CC(C)(C)ON(C=O)CCOc1cc(-c2ccccc2Cl)on1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 9/20 0.38
MEN1 O00255 7/20 0.38
KMT2A Q03164 7/20 0.38
RAB9A P51151 7/20 0.38
CYP1A2 P05177 4/20 0.38
CYP2C19 P33261 4/20 0.38
HPGD P15428 4/20 0.36
ALDH1A1 P00352 2/20 0.36
CYP3A4 P08684 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MAPT P10636 2/20 0.36
NPY1R P25929 1/20 0.36
NPY2R P49146 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KLF5 Q13887 1/20 0.35
CYP2C9 P11712 1/20 0.35
HCRTR1 O43613 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8375001 0.92 NR1H2 (0.31) NPC1MEN1KMT2ARAB9ACYP1A2
SCHEMBL8376904 0.89 ALOX15 (0.36) NPC1MEN1KMT2ARAB9ACYP1A2
SCHEMBL8376838 0.88 NR1H4 (0.32) MEN1KMT2AMAPT
SCHEMBL8377369 0.88 NPC1 (0.34) NPC1MEN1KMT2ARAB9ACYP1A2
SCHEMBL8377399 0.87 ALDH1A1 (0.44) NPC1MEN1KMT2ARAB9AHPGD
SCHEMBL8375699 0.86 SLC6A9 (0.33) NPC1RAB9AHPGDALDH1A1L3MBTL1
SCHEMBL8380161 0.86 NR1H2 (0.36) NPC1KMT2ARAB9ACYP1A2CYP2C19
SCHEMBL8377511 0.85
SCHEMBL8378946 0.85 CXCR1 (0.40) ALDH1A1
SCHEMBL8375024 0.84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6005116-A HAVE INHIBITION ACTIVITIES AGAINST TYPE A-MONOAMINE OXIDASE; TREATING OR PREVENTING DEPRESSION, PARKINSON'S DISEASE, ALZEHEIMER'S DEMENTIA, OR CEREBROVASCULAR DEMENTIA SANKYO COMPANY, LIMITED (JP) 1999-12-21 US disclosed
EP-0885891-A1 ISOXAZOLE DERIVATIVES SANKYO COMPANY LIMITED (JP) 1998-12-23 EP disclosed