SCHEMBL8377369

SCHEMBL8377369

Cc1ccccc1-c1cc(OCCN(C=O)OC(C)(C)C)no1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.34
HPGD P15428 2/20 0.34
RAB9A P51151 2/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
MAPT P10636 1/20 0.34
CYP2C9 P11712 1/20 0.34
NFKB1 P19838 1/20 0.34
CYP2C19 P33261 1/20 0.34
NFKB2 Q00653 1/20 0.34
KMT2A Q03164 1/20 0.34
RELA Q04206 1/20 0.34
ATM Q13315 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ALDH1A1 P00352 1/20 0.32
ALOX15 P16050 1/20 0.32
HSD17B10 Q99714 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8377377 0.88 NPC1 (0.38) NPC1HPGDRAB9AMEN1CYP1A2
SCHEMBL8377399 0.88 ALDH1A1 (0.44) NPC1HPGDRAB9AMEN1MAPT
SCHEMBL8375699 0.87 SLC6A9 (0.33) NPC1HPGDRAB9AMAPTSMN1; SMN2
SCHEMBL8380161 0.87 NR1H2 (0.36) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL8378946 0.86 CXCR1 (0.40) ALDH1A1
SCHEMBL8375001 0.85 NR1H2 (0.31) NPC1RAB9AMEN1CYP1A2CYP2C19
SCHEMBL8375559 0.84 CXCR1 (0.41) NPC1RAB9AALDH1A1
SCHEMBL8375555 0.83 NPC1 (0.35) NPC1HPGDRAB9AMEN1CYP1A2
SCHEMBL8377511 0.82
SCHEMBL8380155 0.81 ACKR3 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6005116-A HAVE INHIBITION ACTIVITIES AGAINST TYPE A-MONOAMINE OXIDASE; TREATING OR PREVENTING DEPRESSION, PARKINSON'S DISEASE, ALZEHEIMER'S DEMENTIA, OR CEREBROVASCULAR DEMENTIA SANKYO COMPANY, LIMITED (JP) 1999-12-21 US disclosed
EP-0885891-A1 ISOXAZOLE DERIVATIVES SANKYO COMPANY LIMITED (JP) 1998-12-23 EP disclosed