SCHEMBL8375800

SCHEMBL8375800

CC(C)c1c(OCCN(C=O)OC(C)(C)C)noc1-c1ccco1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.33
PKM P14618 1/20 0.33
NPC1 O15118 1/20 0.30
TSHR P16473 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8375766 0.85 TSHR (0.31) TSHR
SCHEMBL8377355 0.82 KDM4E (0.32) ALDH1A1NPC1RAB9A
SCHEMBL8375679 0.82 NPC1 (0.31) NPC1RAB9A
SCHEMBL8377411 0.82 TSHR (0.31) TSHR
SCHEMBL8376446 0.81 MAPT (0.31) ALDH1A1NPC1
SCHEMBL8378808 0.81 CHRNB2 (0.33) NPC1RAB9A
SCHEMBL8377392 0.78 PPARD (0.33)
SCHEMBL8377387 0.78 KCNH2 (0.30)
SCHEMBL8377358 0.77 TSHR (0.32) ALDH1A1TSHR
SCHEMBL5618290 0.76 ALDH1A1 (0.38) ALDH1A1PKMNPC1TSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6005116-A HAVE INHIBITION ACTIVITIES AGAINST TYPE A-MONOAMINE OXIDASE; TREATING OR PREVENTING DEPRESSION, PARKINSON'S DISEASE, ALZEHEIMER'S DEMENTIA, OR CEREBROVASCULAR DEMENTIA SANKYO COMPANY, LIMITED (JP) 1999-12-21 US disclosed
EP-0885891-A1 ISOXAZOLE DERIVATIVES SANKYO COMPANY LIMITED (JP) 1998-12-23 EP disclosed