SCHEMBL8377265

SCHEMBL8377265

Oc1cc(-c2ccc(F)cc2)on1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.50
RAB9A P51151 8/20 0.50
MAPT P10636 3/20 0.50
TP53 P04637 2/20 0.50
HTT P42858 2/20 0.50
HDAC6 Q9UBN7 4/20 0.48
PTGS2 P35354 1/20 0.47
TDP1 Q9NUW8 2/20 0.47
KMT2A Q03164 4/20 0.46
MEN1 O00255 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
LMNA P02545 1/20 0.46
HIF1A Q16665 1/20 0.46
ALDH1A1 P00352 1/20 0.44
ASIC1 P78348 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8375802 0.83 ALDH1A1 (0.61) NPC1RAB9AMAPTTP53HDAC6
SCHEMBL6938529 0.80 NOTUM (0.61) NPC1RAB9AMAPTTP53TDP1
SCHEMBL788874 0.80 ALDH1A1 (0.44) NPC1RAB9AMAPTTP53KMT2A
SCHEMBL8380106 0.80 RAB9A (0.57) NPC1RAB9AMAPTPTGS2TDP1
SCHEMBL2959768 0.80 NPC1 (0.56) NPC1RAB9AMAPTTP53HTT
SCHEMBL38657732 0.80 PTPN1 (0.61) NPC1RAB9AMAPTTP53HTT
SCHEMBL8378877 0.79 TRPV1 (0.50) NPC1RAB9AMAPTKMT2AMEN1
SCHEMBL5157687 0.79 RAB9A (0.61) NPC1RAB9AMAPTPTGS2TDP1
SCHEMBL38658113 0.78 ALDH1A1 (0.43) NPC1RAB9ATP53HDAC6TDP1
SCHEMBL21121779 0.78 HSD17B1 (0.64) NPC1RAB9AMAPTTP53HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6005116-A HAVE INHIBITION ACTIVITIES AGAINST TYPE A-MONOAMINE OXIDASE; TREATING OR PREVENTING DEPRESSION, PARKINSON'S DISEASE, ALZEHEIMER'S DEMENTIA, OR CEREBROVASCULAR DEMENTIA SANKYO COMPANY, LIMITED (JP) 1999-12-21 US disclosed
CN-1216986-A Isoxazole derivatives SANKYO CO (JP) 1999-05-19 CN disclosed
EP-0885891-A1 ISOXAZOLE DERIVATIVES SANKYO COMPANY LIMITED (JP) 1998-12-23 EP disclosed