SCHEMBL8377758

SCHEMBL8377758

NC(=NO)c1c(F)ccc(Cl)c1N

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.33
ITGAV P06756 1/20 0.33
PBRM1 Q86U86 1/20 0.31
IDO1 P14902 1/20 0.31
KDM1A O60341 1/20 0.31
CHEK1 O14757 1/20 0.31
NTRK1 P04629 1/20 0.31
PIM1 P11309 1/20 0.31
CDK2 P24941 1/20 0.31
CSNK2A1 P68400 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8376594 0.84 KDM1A (0.34) KDM1A
SCHEMBL8416556 0.79 ITGB3 (0.34) ITGB3ITGAVPBRM1IDO1KDM1A
SCHEMBL7244240 0.79 ITGB3 (0.34) ITGB3ITGAVPBRM1IDO1KDM1A
SCHEMBL8558738 0.79 LMNA (0.39) ITGB3ITGAVPBRM1IDO1
Hydrochloric Acid SCHEMBL8377740 0.77 LMNA (0.42) ITGB3ITGAVIDO1
SCHEMBL7242129 0.76 PBRM1 (0.44) PBRM1
Hydrochloric Acid SCHEMBL8380885 0.76 PBRM1 (0.41) PBRM1IDO1PIM1CDK2CSNK2A1
SCHEMBL2127072 0.73 DPP4 (0.45)
SCHEMBL642255 0.71 CES2 (0.46) KDM1A
SCHEMBL642256 0.71 CES2 (0.46) KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5883102-A Pharmaceutically active compounds ASTRA PHARMACEUTICALS LIMITED (GB) 1999-03-16 US disclosed
EP-0858451-A1 PHARMACEUTICALLY ACTIVE QUINAZOLINE COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-08-19 EP disclosed
WO-1997014686-A1 PHARMACEUTICALLY ACTIVE QUINAZOLINE COMPOUNDS ASTRA PHARMACEUTICALS LIMITED (GB) 1997-04-24 WO disclosed