SCHEMBL8378366

SCHEMBL8378366

NC(=NO)c1c(N)cccc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.40
CES1 P23141 2/20 0.40
KDM1A O60341 4/20 0.36
PREP P48147 1/20 0.36
CRBN Q96SW2 1/20 0.35
CTSL P07711 1/20 0.32
ITGB2 P05107 1/20 0.32
ICAM1 P05362 1/20 0.32
ITGAL P20701 1/20 0.32
GRIN2D O15399 2/20 0.32
GRIN3B O60391 2/20 0.32
GRIN1 Q05586 2/20 0.32
GRIN2A Q12879 2/20 0.32
GRIN2B Q13224 2/20 0.32
GRIN2C Q14957 2/20 0.32
GRIN3A Q8TCU5 2/20 0.32
LMNA P02545 2/20 0.32
ALDH1A1 P00352 1/20 0.31
CYP3A4 P08684 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL642256 0.87 CES2 (0.46) CES2CES1KDM1ACTSLITGB2
SCHEMBL642255 0.87 CES2 (0.46) CES2CES1KDM1ACTSLITGB2
SCHEMBL7242129 0.78 PBRM1 (0.44) CES2CES1ITGB2ICAM1ITGAL
SCHEMBL21163487 0.78 ACHE (0.41) CES2CES1KDM1AGRIN2DGRIN3B
SCHEMBL8381824 0.76 ALDH1A1 (0.43) GRIN2BLMNAALDH1A1CYP3A4TSHR
SCHEMBL6571700 0.76 RORB (0.36) CES2CES1KDM1AGRIN2DGRIN3B
SCHEMBL8376594 0.75 KDM1A (0.34) KDM1A
SCHEMBL164708 0.75 CES2 (0.54) CES2CES1PREPCRBNITGB2
SCHEMBL7952512 0.75 CES2 (0.43) CES2CES1PREPCRBNITGB2
SCHEMBL8381060 0.74 CES2 (0.35) CES2CES1KDM1ACTSLITGB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5883102-A Pharmaceutically active compounds ASTRA PHARMACEUTICALS LIMITED (GB) 1999-03-16 US disclosed