SCHEMBL8380300

SCHEMBL8380300

COCCOc1cc(OC)cc(C#N)c1OCCOC.O=C(CO)OC(c1ccccc1)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
NOS2 P35228 2/20 0.39
RET P07949 3/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HPGD P15428 1/20 0.35
NPC1 O15118 4/20 0.35
RAB9A P51151 4/20 0.35
HSD17B10 Q99714 2/20 0.35
TP53 P04637 1/20 0.35
AR P10275 1/20 0.34
RECQL P46063 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HTR1A P08908 1/20 0.34
ADRA1D P25100 1/20 0.34
ADRA1A P35348 1/20 0.34
ADRA1B P35368 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8378992 0.85 ALDH1A1 (0.39) MEN1KMT2AHPGDALDH1A1HTR1A
Glycolic Acid SCHEMBL8382549 0.83 HPGD (0.46) HPGDNPC1RAB9AHSD17B10TP53
SCHEMBL8636168 0.78 L3MBTL1 (0.47) MEN1KMT2AALDH1A1HTR1AADRA1D
SCHEMBL8378914 0.76 HTR1A (0.39) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL8380298 0.73 HTR1A (0.34) RETHPGDHSD17B10RECQLALDH1A1
SCHEMBL8377272 0.71 HTR1A (0.34) MEN1KMT2AHPGDHSD17B10AR
SCHEMBL8382372 0.69 F2 (0.37) CYP2D6SLC6A2SLC6A4NOS2RET
SCHEMBL7962974 0.69 HPGD (0.36) HPGDNPC1RAB9AHSD17B10TP53
SCHEMBL8378504 0.68 ALDH1A1 (0.34) MEN1KMT2AHPGDHSD17B10RECQL
SCHEMBL7019908 0.68 CRHBP (0.58) CYP2D6KMT2AHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5883248-A QUATERNARY AMMONIUM INTERMEDIATES ROUSSEL UCLAF (FR) 1999-03-16 US disclosed
US-5763617-A Cephalosporins ROUSSEL UCLAF (FR) 1998-06-09 US disclosed
US-5728828-A A 3-(3-CHLORO- OR IODOPROP-1-EN-1-YL),7-(2-AMINOTHIAZOL-4-YL) ((CARBOXY)(PHENYL)METHOXYIMINO)ACETAMIDO-3-CEPHEM; GRAMNEGATIVE AND -POSITIVE BACTERIA, ESP. ANTIBIOTIC-RESISTANCE STAPHYLOCOCCUS ROUSSEL UCLAF (FR) 1998-03-17 US disclosed
US-5712266-A Cephalosporins ROUSSEL UCLAF (FR) 1998-01-27 US disclosed