SCHEMBL8380852

SCHEMBL8380852

CCOC(=O)CN1CCN(C(=O)c2ccc(NC(=N)NC(=O)OC(C)(C)C)cc2)CC1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.43
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.42
NPSR1 Q6W5P4 2/20 0.41
GAA P10253 1/20 0.41
NAMPT P43490 2/20 0.39
ATM Q13315 1/20 0.38
ABL1 P00519 2/20 0.36
RIN1 Q13671 2/20 0.36
EPHX2 P34913 1/20 0.36
ALDH1A1 P00352 4/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
MAPT P10636 2/20 0.36
POLB P06746 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
FLT3 P36888 1/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8384276 0.91 CYP2C19 (0.42) CYP2C19KDM4EHPGDNPSR1GAA
SCHEMBL8385330 0.84 NAMPT (0.40) CYP2C19KDM4EHPGDNAMPTABL1
SCHEMBL8385320 0.80 TGM2 (0.45) KDM4EGAANAMPTMEN1KMT2A
SCHEMBL8380856 0.77 KMT2A (0.36) CYP2C19GAAALDH1A1MEN1KMT2A
SCHEMBL8385474 0.75 ITGB3 (0.45) CYP2C19KDM4EHPGDNPSR1GAA
SCHEMBL8385342 0.69 ITGB3 (0.58) CYP2C19KDM4EHPGDNAMPTMEN1
SCHEMBL8384282 0.69 PLA2G2A (0.36) GAAALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL8385553 0.68 MAPT (0.48) NAMPTEPHX2ALDH1A1MEN1KMT2A
SCHEMBL13017212 0.68 TDP1 (0.44) ALDH1A1MEN1KMT2AMAPTPOLB
SCHEMBL8386317 0.68 EPHX2 (0.41) CYP2C19KDM4EHPGDNPSR1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908843-A Piperazine compounds as fibrinogen inhibitors MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1999-06-01 US disclosed