SCHEMBL8392170

SCHEMBL8392170

N=C(Nc1ccc(CNC(=O)N(c2ccccc2)c2ccccc2)cc1)N1CCCC1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 4/20 0.43
CHRM1 P11229 1/20 0.42
HTR2A P28223 1/20 0.42
MCHR1 Q99705 1/20 0.42
ALDH1A1 P00352 3/20 0.41
MAPT P10636 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
TP53 P04637 1/20 0.41
POLB P06746 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PTPN1 P18031 1/20 0.40
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
RORC P51449 1/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL8392856 0.98 HRH3 (0.42) NAMPTCHRM1HTR2AMCHR1ALDH1A1
SCHEMBL8392136 0.89 GAA (0.46) NAMPTMAPTHRH3SMN1; SMN2ROCK2
SCHEMBL8392369 0.88 POLB (0.41) ALDH1A1MAPTPOLBSMN1; SMN2NPC1
Oxalic Acid SCHEMBL8396187 0.87 GAA (0.44) NAMPTALDH1A1HRH3SMN1; SMN2ROCK2
SCHEMBL8396226 0.80 ALDH1A1 (0.56) NAMPTALDH1A1MAPTTP53ROCK2
SCHEMBL8392174 0.76 TPSAB1 (0.53)
SCHEMBL8393077 0.75 POLB (0.47) NAMPTCHRM1HTR2AMCHR1ALDH1A1
SCHEMBL29221819 0.75 HSP90AA1 (0.53) ALDH1A1MAPTL3MBTL1SMN1; SMN2KMT2A
Bromide SCHEMBL8394207 0.74 POLB (0.46) NAMPTCHRM1HTR2AMCHR1ALDH1A1
SCHEMBL9218989 0.74 MEN1 (0.45) NAMPTALDH1A1MAPTL3MBTL1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0690851-B1 GUANIDINE DERIVATIVES USEFUL IN THERAPY ASTRA AB (SE) 1999-05-19 EP claimed
US-5885985-A Guanidine derivatives useful in therapy ASTRA AKTIEBOLAG (SE) 1999-03-23 US claimed
EP-0690851-A1 GUANIDINE DERIVATIVES USEFUL IN THERAPY Astra Aktiebolag (SE) 1996-01-10 EP claimed
WO-1994021621-A1 GUANIDINE DERIVATIVES USEFUL IN THERAPY ASTRA AKTIEBOLAG (SE) 1994-09-29 WO claimed