SCHEMBL8396226

SCHEMBL8396226

N=C(Nc1ccc(C(=O)NCc2ccccc2)cc1)N1CCCC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.56
NAMPT P43490 5/20 0.53
HDAC2 Q92769 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
MAPT P10636 2/20 0.52
TP53 P04637 1/20 0.52
GAA P10253 1/20 0.52
LMNA P02545 2/20 0.50
ROCK2 O75116 1/20 0.50
RPS6KA5 O75582 1/20 0.50
MAP4K4 O95819 1/20 0.50
PRKCG P05129 1/20 0.50
PRKACA P17612 1/20 0.50
RPS6KB1 P23443 1/20 0.50
MAPK1 P28482 1/20 0.50
AKT1 P31749 1/20 0.50
GSK3A P49840 1/20 0.50
GSK3B P49841 1/20 0.50
PRKX P51817 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8525511 0.88 NAMPT (0.57) NAMPTHDAC2HDAC8HDAC6GAA
SCHEMBL8395852 0.87 MAPK1 (0.55) ALDH1A1HDAC2HDAC8HDAC6TP53
SCHEMBL8524910 0.86 NAMPT (0.64) NAMPTRAB9A
SCHEMBL8523428 0.85 NAMPT (0.60) NAMPTRAB9A
SCHEMBL8392170 0.80 NAMPT (0.43) ALDH1A1NAMPTMAPTTP53ROCK2
Hydrochloric Acid SCHEMBL8582954 0.79 ITGA4 (0.56) ALDH1A1GAALMNAMEN1KMT2A
SCHEMBL17744942 0.78 HDAC6 (0.68) NAMPTHDAC2HDAC8HDAC6MAPT
Oxalic Acid SCHEMBL8392856 0.78 HRH3 (0.42) ALDH1A1NAMPTMAPTTP53ROCK2
SCHEMBL8524903 0.78 NAMPT (0.67) NAMPTMAPTTP53
SCHEMBL22145190 0.76 ALDH1A1 (0.76) ALDH1A1HDAC2HDAC8HDAC6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0690851-B1 GUANIDINE DERIVATIVES USEFUL IN THERAPY ASTRA AB (SE) 1999-05-19 EP claimed
US-5885985-A Guanidine derivatives useful in therapy ASTRA AKTIEBOLAG (SE) 1999-03-23 US claimed