SCHEMBL8399351

SCHEMBL8399351

Fc1cc(F)c2sc(CNc3ccccc3)nc2c1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 8/20 0.46
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TRPM5 Q9NZQ8 1/20 0.36
NOS1 P29475 1/20 0.35
CYP1A2 P05177 1/20 0.35
IDO1 P14902 1/20 0.35
CYP2C19 P33261 1/20 0.35
KCNH3 Q9ULD8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8395489 0.90 AKR1B1 (0.39) AKR1B1NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL8399113 0.89 NOS1 (0.44) AKR1B1NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL8400483 0.86 AKR1B1 (0.44) AKR1B1NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL8395435 0.86 AKR1B1 (0.38) AKR1B1NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL8399262 0.86 AKR1B1 (0.40) AKR1B1NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL8399732 0.86 AKR1B1 (0.42) AKR1B1MAPTRAB9ATRPM5
SCHEMBL8399092 0.86 AKR1B1 (0.38) AKR1B1NOS1
SCHEMBL8395524 0.85 AKR1B1 (0.43) AKR1B1NPC1MAPTRAB9A
SCHEMBL8396655 0.83 HDAC6 (0.50) AKR1B1NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL8396103 0.83 AKR1B1 (0.41) AKR1B1NPC1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647636-B1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF SENJU PHARMA CO (JP) 1999-06-09 EP disclosed
US-5532257-A ENZYME INHIBITOR SENJU PHARMACEUTICAL CO., LTD (JP) 1996-07-02 US disclosed
EP-0647636-A1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Senju Pharmaceutical Co., Ltd. (JP) 1995-04-12 EP disclosed