SCHEMBL8399113

SCHEMBL8399113

Fc1cccc(NCc2nc3cc(F)cc(F)c3s2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.44
HPGD P15428 2/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
TSHR P16473 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
AKR1B1 P15121 6/20 0.40
HDAC6 Q9UBN7 2/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
MAPT P10636 3/20 0.37
KDM4E B2RXH2 1/20 0.37
CCNE1 P24864 1/20 0.36
CDK2 P24941 1/20 0.36
CDK3 Q00526 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8399351 0.89 AKR1B1 (0.46) NOS1NPC1RAB9ASMN1; SMN2AKR1B1
SCHEMBL8399092 0.89 AKR1B1 (0.38) NOS1AKR1B1ERBB2
SCHEMBL8399732 0.89 AKR1B1 (0.42) KMT2AMEN1ALDH1A1RAB9AAKR1B1
SCHEMBL8395489 0.85 AKR1B1 (0.39) KMT2AMEN1NPC1ALDH1A1RAB9A
SCHEMBL8400189 0.85 AKR1B1 (0.36) NOS1AKR1B1
SCHEMBL8399257 0.84 SYK (0.44) KMT2AMEN1NPC1ALDH1A1TSHR
SCHEMBL8396597 0.83 NOS1 (0.43) NOS1HPGDKMT2AMEN1NPC1
SCHEMBL8395435 0.82 AKR1B1 (0.38) KMT2AMEN1NPC1ALDH1A1RAB9A
SCHEMBL8399262 0.82 AKR1B1 (0.40) HPGDKMT2AMEN1NPC1ALDH1A1
SCHEMBL8400483 0.82 AKR1B1 (0.44) HPGDKMT2AMEN1NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647636-B1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF SENJU PHARMA CO (JP) 1999-06-09 EP disclosed
US-5532257-A ENZYME INHIBITOR SENJU PHARMACEUTICAL CO., LTD (JP) 1996-07-02 US disclosed
EP-0647636-A1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Senju Pharmaceutical Co., Ltd. (JP) 1995-04-12 EP disclosed