SCHEMBL8400170

SCHEMBL8400170

Cc1cccc(-c2nsnc2C(=O)O)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.51
KMO O15229 2/20 0.46
MDM2 Q00987 1/20 0.43
DHODH Q02127 2/20 0.42
AKR1C2 P52895 1/20 0.41
AKR1C1 Q04828 1/20 0.41
RXRA P19793 2/20 0.41
RXRB P28702 2/20 0.41
RXRG P48443 2/20 0.41
NR4A2 P43354 1/20 0.41
CSNK1D P48730 1/20 0.41
CSNK1E P49674 1/20 0.41
MAPK14 Q16539 1/20 0.41
TSHR P16473 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
IP6K1 Q92551 1/20 0.40
IP6K3 Q96PC2 1/20 0.40
IP6K2 Q9UHH9 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10338995 0.81 KDM4E (0.52) PIN1DHODHNR4A2TSHRRAB9A
SCHEMBL8397343 0.81 PIN1 (0.50) PIN1KMONR4A2CSNK1D
SCHEMBL8396801 0.81 PIN1 (0.49) PIN1KMOMDM2RXRARXRB
SCHEMBL8396813 0.80 ALPL (0.46) DHODHMEN1KMT2ACNR1RAB9A
SCHEMBL8400098 0.78 PIN1 (0.52) PIN1KMONPSR1IP6K1IP6K3
SCHEMBL2057011 0.76 KMO (0.52) PIN1KMOMDM2DHODHAKR1C2
SCHEMBL2988256 0.74 RAB9A (0.38) PIN1KMORXRARXRBRXRG
SCHEMBL11400729 0.74 AKR1C2 (0.47) PIN1KMODHODHAKR1C2AKR1C1
SCHEMBL11390925 0.73 KMO (0.43) PIN1KMODHODHAKR1C2AKR1C1
SCHEMBL11005057 0.72 AKR1C2 (0.45) PIN1KMOMDM2DHODHAKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5948916-A Arylthiadiazole derivative and antiviral agent containing the same RATIONAL DRUG DESIGN LABORATORIES (JP) 1999-09-07 US disclosed
EP-0785193-A1 ARYLTHIADIAZOLE DERIVATIVE AND ANTIVIRAL AGENT CONTAINING THE SAME Rational Drug Design Laboratories (JP) 1997-07-23 EP disclosed