SCHEMBL8401940

SCHEMBL8401940

CN(Cc1cnc(Br)s1)C(=C[N+](=O)[O-])NCCF

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.31
PDK1 Q15118 1/20 0.31
PDK2 Q15119 1/20 0.31
PDK3 Q15120 1/20 0.31
PDK4 Q16654 1/20 0.31
MEN1 O00255 1/20 0.30
SLC22A1 O15245 1/20 0.30
ABCB11 O95342 1/20 0.30
LMNA P02545 1/20 0.30
CHRM2 P08172 1/20 0.30
CHRM1 P11229 1/20 0.30
TSHR P16473 1/20 0.30
ADRA2C P18825 1/20 0.30
NFKB1 P19838 1/20 0.30
CHRM3 P20309 1/20 0.30
ATP4A P20648 1/20 0.30
PTGS1 P23219 1/20 0.30
HRH2 P25021 1/20 0.30
SLC6A4 P31645 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8404109 0.89 RECQL (0.35) ACHEMEN1SLC22A1ABCB11LMNA
SCHEMBL8698690 0.87 PDK1 (0.32) ACHEPDK1PDK2PDK3PDK4
SCHEMBL7664952 0.85 ACHE (0.33) ACHEPDK1PDK2PDK3PDK4
SCHEMBL8405612 0.83 PDK1 (0.32) PDK1PDK2PDK3PDK4
SCHEMBL8401805 0.79 MMP2 (0.35) ACHEMEN1SLC22A1ABCB11LMNA
SCHEMBL7662711 0.78
SCHEMBL7664910 0.77 PDK1 (0.36) PDK1PDK2PDK3PDK4
SCHEMBL8401724 0.76 RECQL (0.36) ACHEMEN1LMNAKMT2AMAPT
SCHEMBL8401739 0.75 RECQL (0.36) MEN1LMNAKMT2AMAPT
SCHEMBL7662506 0.74 PDK1 (0.32) PDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5935981-A INSECTICIDAL/MITICIDAL ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-08-10 US disclosed
US-5849768-A α-unsaturated amines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-12-15 US disclosed