SCHEMBL8409543

SCHEMBL8409543

COC(=O)CC1CCCN(c2ccc(-c3ccc(C#N)cc3)c(C)c2)C1

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 14/20 0.41
USP14 P54578 1/20 0.41
HRH2 P25021 1/20 0.39
HRH1 P35367 1/20 0.39
CHRM3 P20309 1/20 0.39
LRRK2 Q5S007 1/20 0.38
NLRP3 Q96P20 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8409450 0.95 KDM1A (0.40) KDM1AHRH2HRH1
SCHEMBL8407654 0.89 HRH2 (0.41) KDM1AUSP14HRH2HRH1
SCHEMBL8407178 0.86 KDM1A (0.38) KDM1AUSP14CHRM3LRRK2
SCHEMBL8407652 0.83 HRH2 (0.45) KDM1AHRH2HRH1
SCHEMBL8407515 0.81 KDM1A (0.38) KDM1A
SCHEMBL8409141 0.79 USP14 (0.46) KDM1AUSP14HRH2HRH1CHRM3
SCHEMBL8715693 0.79 KDM1A (0.42) KDM1ALRRK2
SCHEMBL5535336 0.76 KDM4E (0.39) KDM1AUSP14
SCHEMBL8718962 0.76 CHRM4 (0.38) KDM1A
SCHEMBL5526338 0.75 NOTUM (0.59)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5922763-A ANTICOAGULANT; CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1999-07-13 US disclosed
US-5736559-A CARDIOVASCULAR DISORDERS; RESPIRATORY SYSTEM DISORDERS KARL THOMAE GMBH (DE) 1998-04-07 US disclosed