SCHEMBL8410474

SCHEMBL8410474

N=C(N)c1ccc(-c2ccc(CCN3CCC(C(=O)O)CC3)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.53
HTR2C P28335 2/20 0.53
HTR7 P34969 2/20 0.53
HTR6 P50406 2/20 0.53
ITGB3 P05106 5/20 0.49
ITGA2B P08514 5/20 0.49
HRH3 Q9Y5N1 2/20 0.49
PRSS1 P07477 2/20 0.46
PRSS2 P07478 2/20 0.46
PRSS3 P35030 2/20 0.46
KCNH2 Q12809 1/20 0.45
LTA4H P09960 1/20 0.44
OPRM1 P35372 1/20 0.44
F2 P00734 1/20 0.43
PLG P00747 1/20 0.43
ST14 Q9Y5Y6 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8410661 0.86 SLC6A1 (0.48) ITGB3ITGA2BHRH3
Hydrochloric Acid SCHEMBL8407181 0.85 THRA (0.54) HTR2AHTR2CHTR7HTR6HRH3
SCHEMBL8410297 0.81 ITGB3 (0.52) ITGB3ITGA2BHRH3LTA4H
SCHEMBL8491424 0.80 HTR2A (0.57) HTR2AHTR2CHTR7HTR6HRH3
Hydrochloric Acid SCHEMBL8407670 0.79 L3MBTL1 (0.61) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL1519356 0.78 HTR2A (0.75) HTR2ALTA4HOPRM1
SCHEMBL18117071 0.77 KCNH2 (0.59) HTR2AHTR2CHTR7HTR6HRH3
SCHEMBL4227924 0.77 HTR2A (0.74) HTR2AHTR2CHTR7HTR6
SCHEMBL15566801 0.77 HTR2A (0.57) HTR2AHTR2CHTR7HTR6HRH3
SCHEMBL8407585 0.77 CHRNB2 (0.49) ITGB3ITGA2BHRH3LTA4HF2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5922763-A ANTICOAGULANT; CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1999-07-13 US disclosed
US-5736559-A CARDIOVASCULAR DISORDERS; RESPIRATORY SYSTEM DISORDERS KARL THOMAE GMBH (DE) 1998-04-07 US disclosed
US-5597825-A AGGREGATION INHIBITORS DR. KARL THOMAE GMBH (DE) 1997-01-28 US disclosed
EP-0496378-A1 Biphenylderivatives, drugs containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1992-07-29 EP disclosed