SCHEMBL8416384

SCHEMBL8416384

CNc1cc(NS(=O)(=O)c2cc[c]cc2)nc(N2CCCC2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 0.48
MAPT P10636 3/20 0.47
ALDH1A1 P00352 3/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
RAB9A P51151 1/20 0.47
KDM4E B2RXH2 1/20 0.46
APEX1 P27695 1/20 0.46
BLM P54132 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
KMO O15229 5/20 0.41
GALR2 O43603 2/20 0.39
NUDT1 P36639 2/20 0.37
RECQL P46063 1/20 0.36
HSD11B1 P28845 1/20 0.36
GALR1 P47211 1/20 0.36
MEN1 O00255 1/20 0.35
GAA P10253 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7823458 0.85 HTR6 (0.68) HTR6MAPTALDH1A1CYP3A4CYP2C9
SCHEMBL8416375 0.85 GAA (0.37) MAPTALDH1A1KMOGALR2RECQL
SCHEMBL7823536 0.83 HTR6 (0.68) HTR6MAPTALDH1A1CYP3A4CYP2C9
SCHEMBL7836309 0.81 GFER (0.58) MAPTALDH1A1KDM4EMEN1GAA
SCHEMBL7832160 0.71 L3MBTL1 (0.53) HTR6MAPTALDH1A1CYP3A4CYP2C9
SCHEMBL8413208 0.69 HTR6 (0.54) HTR6MAPTALDH1A1CYP3A4CYP2C9
SCHEMBL7838498 0.68 GFER (0.57) MAPTALDH1A1KDM4ENPSR1MEN1
SCHEMBL7833289 0.68 LMNA (0.50) HTR6MAPTALDH1A1CYP3A4CYP2C9
SCHEMBL11757838 0.68 PDE4A (0.69) ALDH1A1KDM4EHSD11B1MEN1KMT2A
SCHEMBL9217636 0.68 NUDT1 (0.68) MAPTALDH1A1KDM4EBLMNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939451-A INDOL-4-YL-BENZENESULFONAMIDES AS ACTIVE MATERIAL TREATING MALARIA, BACTERIAL INFECTION, NEUROLOGICAL DISORDERS HOFFMANN-LA ROCHE INC. (US) 1999-08-17 US disclosed
US-5932599-A 4-AMINO-N-(PYRIDINYL-4-YL)-BENZENESULFONAMIDES AS ACTIVE MATERIAL TREATING MALARIA, BACTERIAL INFECTION, NEUROLOGICAL DISORDERS HOFFMANN-LA ROCHE INC. (US) 1999-08-03 US disclosed