SCHEMBL8418644

SCHEMBL8418644

ICCCc1nnnn1C(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DAGLA Q9Y4D2 2/20 0.35
NPSR1 Q6W5P4 3/20 0.33
LMNA P02545 2/20 0.33
AGTR1 P30556 1/20 0.32
AGTR2 P50052 1/20 0.32
HSD11B1 P28845 6/20 0.32
HTT P42858 2/20 0.31
PKM P14618 1/20 0.31
NLRP3 Q96P20 1/20 0.31
ALDH1A1 P00352 2/20 0.31
POLB P06746 1/20 0.31
MEN1 O00255 1/20 0.30
TSHR P16473 1/20 0.30
KMT2A Q03164 1/20 0.30
APEX1 P27695 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8417361 0.95 DAGLA (0.34) DAGLANPSR1LMNAAGTR1AGTR2
SCHEMBL7202719 0.85 DAGLA (0.35) DAGLANPSR1LMNAAGTR1AGTR2
SCHEMBL838908 0.85 SLC9A1 (0.36) DAGLANPSR1LMNAAGTR1AGTR2
SCHEMBL5357964 0.84 LMNA (0.35) NPSR1LMNAAGTR1AGTR2HSD11B1
SCHEMBL3568399 0.84 SLC9A1 (0.35) DAGLANPSR1LMNAAGTR1AGTR2
SCHEMBL14032263 0.81 AGTR1 (0.35) DAGLANPSR1LMNAAGTR1AGTR2
SCHEMBL3260686 0.81 CYP2A6 (0.34) NPSR1LMNAAGTR1AGTR2HSD11B1
SCHEMBL22615880 0.81 HSD11B1 (0.36) DAGLANPSR1LMNAAGTR1AGTR2
SCHEMBL2970884 0.80 LMNA (0.36) DAGLANPSR1LMNAHTTALDH1A1
SCHEMBL2359649 0.78 LMNA (0.35) NPSR1LMNAAGTR1AGTR2HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0684257-B1 Pseudopeptide derivatives of neurokinines, process for their preparation and pharmaceutical compositions comprising them ADIR (FR) 1999-09-22 EP disclosed
US-5561113-A ANALGESICS; ANTIIFLAMMATORY AGENTS; GASTROINTESTINAL, UROGENITAL AND NERVOUS SYSTEM(CNS) DISORDERS; ASTHMA; ANTIALLERGENS ADIR ET COMPAGNIE (FR) 1996-10-01 US disclosed
EP-0684257-A1 Pseudopeptide derivatives of neurokinines, process for their preparation and pharmaceutical compositions comprising them ADIR ET COMPAGNIE (FR) 1995-11-29 EP disclosed