SCHEMBL8419864

SCHEMBL8419864

C=CCOc1ccc(CC(C)(C)C(=O)OC)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.46
ADRB2 P07550 1/20 0.45
ADRB1 P08588 1/20 0.45
ADRB3 P13945 1/20 0.45
NPC1 O15118 4/20 0.45
MAPT P10636 3/20 0.45
RAB9A P51151 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
POLB P06746 2/20 0.45
ALDH1A1 P00352 2/20 0.45
USP2 O75604 1/20 0.45
CACNA1B Q00975 1/20 0.45
APBA1 Q02410 1/20 0.45
BLM P54132 1/20 0.42
CHRNB2 P17787 3/20 0.42
CHRNB4 P30926 3/20 0.42
CHRNA3 P32297 3/20 0.42
CHRNA4 P43681 3/20 0.42
KDM4E B2RXH2 1/20 0.41
CA12 O43570 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11509018 0.81 PTPRB (0.47) BLMCA1CA2
SCHEMBL13903099 0.80 PTPRB (0.54) NPC1RAB9ASMN1; SMN2ALDH1A1CA1
SCHEMBL3180737 0.79 SMN1; SMN2 (0.50) ADRB2ADRB1ADRB3NPC1MAPT
SCHEMBL4456470 0.78 ALDH1A1 (0.50) FFAR1ADRB2ADRB1ADRB3NPC1
SCHEMBL13085360 0.78 ADRB2 (0.44) FFAR1ADRB2ADRB1ADRB3NPC1
SCHEMBL3656838 0.77 NPC1 (0.56) FFAR1NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL9023615 0.77 PTPRB (0.42) ALDH1A1BLMCA1CA2
SCHEMBL9575627 0.77 MAPT (0.47) FFAR1ADRB2ADRB1ADRB3NPC1
SCHEMBL11646444 0.76 PTPRB (0.44) BLM
SCHEMBL13903112 0.76 LTA4H (0.48) MAPTSMN1; SMN2ALDH1A1KDM4ECYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919793-A QUINUCLIDINE DERIVATIVES, SQUALENE SYNTHETASE INHIBITORS, ANTICHOLESTEROL AGENTS ZENECA LIMITED (GB) 1999-07-06 US disclosed
CN-1121718-A Heterocyclic derivatives ZENECA LTD (GB) 1996-05-01 CN disclosed
EP-0696284-A1 HETEROCYCLIC DERIVATIVES ZENECA LIMITED (GB) 1996-02-14 EP disclosed
WO-1994025459-A1 HETEROCYCLIC DERIVATIVES ZENECA LIMITED (GB) 1994-11-10 WO disclosed