SCHEMBL8425248

SCHEMBL8425248

CC(=O)NC1(c2ccccc2)CCN(CCCCn2cnnc2-c2ccccc2)CC1c1ccc(Cl)c(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 17/20 0.40
TACR2 P21452 3/20 0.40
TACR1 P25103 2/20 0.40
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8425245 0.82 ADRA1D (0.39) TACR3TACR2TACR1ADRA2AADRA2B
SCHEMBL6160860 0.74 TACR2 (0.62) TACR3TACR2TACR1
Hydrochloric Acid SCHEMBL8425489 0.70 ADRA2A (0.36) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL8425178 0.69 ALDH1A1 (0.36) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL8425278 0.69 P2RX7 (0.43) ADRA2AADRA2BADRA2CADRA1DADRA1A
Hydrochloric Acid SCHEMBL6161088 0.63 TACR2 (0.61) TACR3TACR2TACR1
Hydrochloric Acid SCHEMBL7988071 0.63 TACR2 (0.61) TACR3TACR2TACR1
SCHEMBL2478765 0.62 TACR3 (0.53) TACR3TACR2TACR1
SCHEMBL2480008 0.62 TACR3 (0.50) TACR3TACR2TACR1
Hydrochloric Acid SCHEMBL8364985 0.62 TACR3 (0.46) TACR3TACR2TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5889024-A Substituted heterocycles ZENECA LIMITED (GB) 1999-03-30 US disclosed