SCHEMBL8425910

SCHEMBL8425910

[CH2]C(C)(OP(=O)(O)Cc1ccccc1)c1cccnc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 1/20 0.46
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HIF1A Q16665 1/20 0.43
FDPS P14324 7/20 0.42
LMNA P02545 2/20 0.42
BTN3A1 O00481 1/20 0.42
PDE3A Q14432 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
GPR132 Q9UNW8 1/20 0.40
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
ANPEP P15144 1/20 0.38
ERAP2 Q6P179 1/20 0.38
ERAP1 Q9NZ08 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7605187 0.85 FDPS (0.45) KCNA5CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL5054253 0.81 KCNA5 (0.40) KCNA5CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7614098 0.81 FDPS (0.43) KCNA5CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7606737 0.79 FDPS (0.42) KCNA5CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7605932 0.78 PTPN1 (0.52) CYP3A4
SCHEMBL8423445 0.77 PGK1 (0.33) FDPS
SCHEMBL7610589 0.76 ALDH1A1 (0.44) FDPSALDH1A1
SCHEMBL7612297 0.74 FDPS (0.47) KCNA5CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7772647 0.74 HPGD (0.46) FDPS
SCHEMBL7609429 0.73 FDPS (0.46) KCNA5CYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0949922-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING COMPULSIVE DISORDERS USING NAALADASE INHIBITORS GUILFORD PHARMACEUTICALS INC. (US) 1999-10-20 EP disclosed
WO-1998013044-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF TREATING COMPULSIVE DISORDERS USING NAALADASE INHIBITORS GUILFORD PHARMACEUTICALS INC. (US) 1998-04-02 WO disclosed