SCHEMBL8428396

SCHEMBL8428396

COc1ccc([C@H](C)N=Cc2cncs2)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 5/20 0.44
CYP19A1 P11511 6/20 0.41
CYP11B2 P19099 2/20 0.41
SLC6A4 P31645 1/20 0.41
ALDH1A1 P00352 2/20 0.34
MAPT P10636 2/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34
HTT P42858 1/20 0.34
NPBWR1 P48145 2/20 0.34
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33
CYP17A1 P05093 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
MCHR1 Q99705 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8428702 0.72 CTH (0.42) SLC6A3CYP19A1ALDH1A1MAPTKDM4E
SCHEMBL8428699 0.72 CTH (0.42) SLC6A3CYP19A1ALDH1A1MAPTKDM4E
SCHEMBL8426401 0.70 TRPA1 (0.50) ALDH1A1MAPTKDM4EGAATDP1
SCHEMBL8426400 0.70 TRPA1 (0.50) ALDH1A1MAPTKDM4EGAATDP1
SCHEMBL19076193 0.70 CYP1A2 (0.56) CYP19A1CYP11B2ALDH1A1MAPTKDM4E
SCHEMBL8428337 0.69 TP53 (0.47) ALDH1A1MAPTGAAHTTTSHR
SCHEMBL28461031 0.68
SCHEMBL16478537 0.68 RAB9A (0.45) ALDH1A1MAPTKDM4ELMNAGAA
SCHEMBL7592948 0.67 TRPA1 (0.50) ALDH1A1MAPTKDM4EGAATDP1
SCHEMBL7592950 0.67 TRPA1 (0.50) ALDH1A1MAPTKDM4EGAATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939561-A Process for the preparation of β-phenylisoserine and β-lactam and their analogues RHONE-POULENCE RORER S.A. (FR) 1999-08-17 US disclosed