SCHEMBL8428869

SCHEMBL8428869

CCCC(=O)OS(=O)(=O)c1ccc(-c2cccc(NC(=N)N)c2)cc1NC=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.34
PAX8 Q06710 2/20 0.33
F2R P25116 1/20 0.33
MAP4K4 O95819 2/20 0.33
ITGB3 P05106 4/20 0.33
ITGAV P06756 4/20 0.33
F10 P00742 1/20 0.33
HDAC6 Q9UBN7 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPK1 P28482 1/20 0.32
PTPN1 P18031 1/20 0.32
PTPRA P18433 1/20 0.32
USP2 O75604 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8430895 0.76 DHODH (0.41) DHODHPAX8ITGB3ITGAVF10
SCHEMBL8429036 0.72 DHODH (0.51) DHODHPAX8ITGB3ITGAVF10
SCHEMBL8432249 0.72 CYP17A1 (0.35) DHODHPAX8ITGB3ITGAVHDAC6
SCHEMBL8432423 0.67 DHODH (0.40) DHODHPAX8ITGB3ITGAVALDH1A1
SCHEMBL8542542 0.67 ITGB3 (0.39) DHODHPAX8ITGB3ITGAVALDH1A1
SCHEMBL27113200 0.65 CYP3A4 (0.54) MAP4K4ALDH1A1MAPK1HPGDSMN1; SMN2
SCHEMBL8409079 0.65 HDAC6 (0.54) HDAC6
SCHEMBL27115412 0.64 TERT (0.49) F2RMAP4K4HDAC6CYP3A4CYP2D6
SCHEMBL8432464 0.64 DHODH (0.43) DHODHITGB3ITGAVF10
SCHEMBL8409081 0.62 LMNA (0.46) ITGB3HDAC6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US disclosed