SCHEMBL8430895

SCHEMBL8430895

CCOC(=O)CCc1ccc(-c2cccc(NC(=N)N)c2)cc1NC=O

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.41
SYK P43405 5/20 0.38
CYP4F2 P78329 1/20 0.37
CYP4A11 Q02928 1/20 0.37
EGFR P00533 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
F9 P00740 1/20 0.35
F10 P00742 1/20 0.35
PARP14 Q460N5 1/20 0.34
PAX8 Q06710 1/20 0.34
MGLL Q99685 1/20 0.34
ITGB3 P05106 1/20 0.34
ITGAV P06756 1/20 0.34
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8432423 0.92 DHODH (0.40) DHODHSYKCYP4F2CYP4A11ALDH1A1
SCHEMBL8430846 0.86 F10 (0.41) CYP4F2CYP4A11ALDH1A1GAAF9
SCHEMBL8429036 0.79 DHODH (0.51) DHODHGAAF10PAX8MGLL
SCHEMBL8428869 0.76 DHODH (0.34) DHODHALDH1A1F10PAX8ITGB3
SCHEMBL8532684 0.73 ENPP2 (0.35) DHODHSYKCYP4F2CYP4A11ALDH1A1
SCHEMBL8432817 0.72 CYP17A1 (0.33)
SCHEMBL8432249 0.71 CYP17A1 (0.35) DHODHPAX8ITGB3ITGAV
SCHEMBL8432464 0.71 DHODH (0.43) DHODHF10MGLLITGB3ITGAV
SCHEMBL8430854 0.70 DHODH (0.43) DHODHALDH1A1F10MGLLITGB3
SCHEMBL8432812 0.70 ITGB3 (0.39) PAX8ITGB3ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US disclosed