SCHEMBL8429031

SCHEMBL8429031

CC(C)CC(=O)N(NC=O)[C@@H](Cc1ccccc1)C(=O)Oc1cc(NC(=N)N)cc(C(F)(F)F)c1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.35
TRPA1 O75762 2/20 0.34
PPARG P37231 1/20 0.34
PPARA Q07869 1/20 0.34
UBE2M P61081 10/20 0.34
DCUN1D1 Q96GG9 10/20 0.34
PDK1 Q15118 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33
SCN9A Q15858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8429203 0.91 TACR1 (0.33) TACR1TRPA1PPARGPPARAUBE2M
SCHEMBL8429038 0.91 TACR1 (0.34) TACR1TRPA1PPARGPPARAUBE2M
SCHEMBL8429096 0.81 UBE2M (0.38) TACR1TRPA1PPARGPPARAUBE2M
SCHEMBL8430965 0.79 PDK1 (0.36) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL8429153 0.77 SIRT2 (0.37) ALDH1A1
SCHEMBL8431034 0.77 ALDH1A1 (0.41) UBE2MDCUN1D1ALDH1A1
SCHEMBL8431230 0.76 RAB9A (0.40) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL8430957 0.76 PLAU (0.38) UBE2MDCUN1D1ALDH1A1
SCHEMBL8429053 0.76 BACE1 (0.36) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL8428894 0.76 BACE1 (0.36) PDK1PDK2PDK3PDK4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US claimed