SCHEMBL8429038

SCHEMBL8429038

CC(C)COC(=O)N(NC=O)[C@@H](Cc1ccccc1)C(=O)Oc1cc(NC(=N)N)cc(C(F)(F)F)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 5/20 0.34
UBE2M P61081 6/20 0.33
DCUN1D1 Q96GG9 6/20 0.33
CACNA1F O60840 2/20 0.33
CACNA1D Q01668 2/20 0.33
CACNA1S Q13698 2/20 0.33
CACNA1C Q13936 2/20 0.33
SCN9A Q15858 1/20 0.33
TRPA1 O75762 1/20 0.33
PPARG P37231 1/20 0.33
PPARA Q07869 1/20 0.33
USP2 O75604 2/20 0.33
CYP3A4 P08684 2/20 0.33
NR1I2 O75469 1/20 0.33
ADRB1 P08588 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8429031 0.91 TACR1 (0.35) TACR1UBE2MDCUN1D1SCN9ATRPA1
SCHEMBL8429153 0.87 SIRT2 (0.37) USP2
SCHEMBL8429203 0.87 TACR1 (0.33) TACR1UBE2MDCUN1D1TRPA1PPARG
SCHEMBL8429096 0.80 UBE2M (0.38) TACR1UBE2MDCUN1D1TRPA1PPARG
SCHEMBL8431034 0.79 ALDH1A1 (0.41) UBE2MDCUN1D1USP2
SCHEMBL7375612 0.79 TRPA1 (0.38) TACR1UBE2MDCUN1D1TRPA1USP2
SCHEMBL7375074 0.79 TRPA1 (0.38) TACR1UBE2MDCUN1D1TRPA1USP2
SCHEMBL8431230 0.79 RAB9A (0.40) USP2ADRB1
SCHEMBL8430957 0.78 PLAU (0.38) UBE2MDCUN1D1USP2
SCHEMBL8432438 0.78 RAB9A (0.37) USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US claimed
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US disclosed