SCHEMBL8429052

SCHEMBL8429052

NN=CNc1cccc([C@@](C(=O)O)(C(=C=O)c2ccccc2)N(N)S(=O)(=O)C=Cc2ccccc2)c1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.34
KMT2A Q03164 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA4 P22748 1/20 0.31
MAOB P27338 1/20 0.31
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8429290 0.86 CA1 (0.33) KMT2ACA1CA2CA4
SCHEMBL8430880 0.85 CA1 (0.37) KMT2ACA1CA2CA4
SCHEMBL8431435 0.82 CA1 (0.32) KMT2ACA1CA2CA4
SCHEMBL8430809 0.81 CA1 (0.32) KMT2ACA1CA2CA4
SCHEMBL8431176 0.81 UBE2M (0.34) CA1CA2CA4
SCHEMBL8431235 0.80 RXFP1 (0.32) KMT2ACA1CA2CA4
SCHEMBL8430969 0.79 NR1H4 (0.33) PPARGKMT2A
SCHEMBL8429055 0.78 TRPV4 (0.35) PPARGKMT2ACA1CA2CA4
SCHEMBL8432441 0.78 KMT2A (0.32) KMT2ACA1CA2CA4
SCHEMBL8430960 0.77 MAPT (0.35) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US claimed
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US disclosed